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结果 1-4(共 4 条),针对检索条件:ALLNAMES:(Matulis) 专利局:all 语言:zh 词根提取:false
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标题Ctr公布日
申请号申请人发明人国际分类
5-ARYL-4-(5-SUBSTITUTED 2,4-DIHYDROXYPHENYL)-1,2,3-THIADIAZOLES AS INHIBITORS OF HSP90 CHAPERONE AND THE INTERMEDIATES FOR PRODUCTION THEREOF
WO05.11.2009
PCT/LT2008/000003BIOTECHNOLOGIJOS INSTITUTASMATULIS, Daumantas
C07D 285/06
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
285
Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/-C07D283/183
01
Five-membered rings
02
Thiadiazoles; Hydrogenated thiadiazoles
04
not condensed with other rings
06
1,2,3-Thiadiazoles; Hydrogenated 1,2,3-thiadiazoles
Invention is related to novel compounds - 5-aryl-4-(5-substituted 2,4-dihydroxyphenyl)-1,2,3-thiadiazoles with general formula (I). The compounds can be used in biomedicine as active ingredients in pharmaceutical formulations, because they inhibit Hsp90 chaperone which participate in cancer progression. This invention is also related to new intermediate compounds which are used for the synthesis of thiadiazoles of general formula (I).

BENZIMIDAZO[1,2-C][1,2,3]THIADIAZOL-7-SULFONSÄUREAMIDE ALS CARBOANHYDRASEINHIBITOREN UND ZWISCHENPRODUKTE ZU DEREN HERSTELLUNG
EP06.05.2009
07793796BIOTECHNOLOGIJOS INSTMATULIS DAUMANTAS
C07D 513/04
C 化学;冶金
07
有机化学
D
杂环化合物(高分子化合物入C08)
513
杂环化合物,在稠环系中至少有1个杂环具有氮原子和硫原子作为仅有的杂环原子,不包含在C07D 463/00、C07D 477/00或C07D 499/00至C07D 507/00组中
02
稠环系中含有两个杂环
04
邻位稠合系
The invention is related to novel compounds - benzimidazo[1,2-c][1,2,3]thiadiazole sulfonamides, corresponding to the general formula (I). The compounds can be used in biomedicine as active ingredients in pharmaceutical formulations, because they inhibit enzymes which participate in disease progression such as glaucome. The compounds of formula (I) inhibits enzymes such as carbonic anhydrases and metallo proteinases. This invention is also related to new intermediate compounds which are used for the synthesis of sulfonamides of formula (I).

5-ARYL-4-(5-SUBSTITUTED 2,4-DIHYDROXYFENIL)-1,2,3-THIADIAZOLES AS INHIBITORS OF HSP90 CHAPERONE AND THE INTERMEDIATES FOR PRODUCTION THEREOF
LT25.11.2009
2008035BIOTECHNOLOGIJOS INSTMATULIS DAUMANTAS
C07D 285/00
C 化学;冶金
07
有机化学
D
杂环化合物(高分子化合物入C08)
285
杂环化合物,有氮原子和硫原子作为仅有的杂环原子的环,不包含在C07D 275/00至C07D 283/00组中
Ivention is related to novel compounds - 5-aryl-4-(5-substituted 2,4-dihydroxyphenyl)-1,2,3-thiadiazoles with general formula (I). The compounds can be used in biomedicine as active ingredients in pharmaceutical formulations, because they inhibit Hsp90 chaperone which participate in cancer progression. This invention is also related to new intermediate compounds which are used for the synthesis of thiadiazoles of formula (I).@

BENZIMIDAZO[1,2-C][1,2,3]THIADIAZOL-7-SULFONSÄUREAMIDE ALS CARBOANHYDRASEINHIBITOREN UND ZWISCHENPRODUKTE ZU DEREN HERSTELLUNG
EP06.05.2009
07793796BIOTECHNOLOGIJOS INSTMATULIS DAUMANTAS
C07D 513/04
C 化学;冶金
07
有机化学
D
杂环化合物(高分子化合物入C08)
513
杂环化合物,在稠环系中至少有1个杂环具有氮原子和硫原子作为仅有的杂环原子,不包含在C07D 463/00、C07D 477/00或C07D 499/00至C07D 507/00组中
02
稠环系中含有两个杂环
04
邻位稠合系
The invention is related to novel compounds - benzimidazo[1,2-c][1,2,3]thiadiazole sulfonamides, corresponding to the general formula (I). The compounds can be used in biomedicine as active ingredients in pharmaceutical formulations, because they inhibit enzymes which participate in disease progression such as glaucome. The compounds of formula (I) inhibits enzymes such as carbonic anhydrases and metallo proteinases. This invention is also related to new intermediate compounds which are used for the synthesis of sulfonamides of formula (I).

结果 1-4(共 4 条),针对检索条件:ALLNAMES:(Matulis) 专利局:all 语言:zh 词根提取:false
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