Traitement en cours

Veuillez attendre...

PATENTSCOPE sera indisponible durant quelques heures pour des raisons de maintenance le dimanche 05.04.2020 à 10:00 AM CEST
Paramétrages

Paramétrages

1. WO2005002626 - COMPOSES DE PHOSPHONATE THERAPEUTIQUES

Numéro de publication WO/2005/002626
Date de publication 13.01.2005
N° de la demande internationale PCT/US2004/013283
Date du dépôt international 26.04.2004
Demande présentée en vertu du Chapitre 2 08.11.2004
CIB
A61K 47/48 2006.01
ANÉCESSITÉS COURANTES DE LA VIE
61SCIENCES MÉDICALE OU VÉTÉRINAIRE; HYGIÈNE
KPRÉPARATIONS À USAGE MÉDICAL, DENTAIRE OU POUR LA TOILETTE
47Préparations médicinales caractérisées par les ingrédients non actifs utilisés, p.ex. les supports ou les additifs inertes; Agents de ciblage ou de modification chimiquement liés à l’ingrédient actif
48l'ingrédient non actif étant chimiquement lié à l'ingrédient actif, p.ex. conjugués polymère-médicament
C07F 9/02 2006.01
CCHIMIE; MÉTALLURGIE
07CHIMIE ORGANIQUE
FCOMPOSÉS ACYCLIQUES, CARBOCYCLIQUES OU HÉTÉROCYCLIQUES CONTENANT DES ÉLÉMENTS AUTRES QUE LE CARBONE, L'HYDROGÈNE, LES HALOGÈNES, L'OXYGÈNE, L'AZOTE, LE SOUFRE, LE SÉLÉNIUM OU LE TELLURE
9Composés contenant des éléments des groupes 5 ou 15 de la classification périodique
02Composés du phosphore
CPC
C07F 9/4006
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
9Compounds containing elements of Groups 5 or 15 of the Periodic System
02Phosphorus compounds
28with one or more P—C bonds
38Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids ; , i.e. RP(=X)(XH)2 (X = S, Se)
40Esters thereof
4003the acid moiety containing a substituent or a structure which is considered as characteristic
4006Esters of acyclic acids which can have further substituents on alkyl
C07F 9/4465
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
9Compounds containing elements of Groups 5 or 15 of the Periodic System
02Phosphorus compounds
28with one or more P—C bonds
38Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids ; , i.e. RP(=X)(XH)2 (X = S, Se)
44Amides thereof
4461the amide moiety containing a substituent or a structure which is considered as characteristic
4465of aliphatic amines
C07F 9/5304
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
9Compounds containing elements of Groups 5 or 15 of the Periodic System
02Phosphorus compounds
28with one or more P—C bonds
50Organo-phosphines
53Organo-phosphine oxides; Organo-phosphine thioxides
5304Acyclic saturated phosphine oxides or thioxides
C07F 9/650952
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
9Compounds containing elements of Groups 5 or 15 of the Periodic System
02Phosphorus compounds
547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
645having two nitrogen atoms as the only ring hetero atoms
6509Six-membered rings
650952having the nitrogen atoms in the positions 1 and 4
C07F 9/653
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
9Compounds containing elements of Groups 5 or 15 of the Periodic System
02Phosphorus compounds
547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
6527having nitrogen and oxygen atoms as the only ring hetero atoms
653Five-membered rings
C07F 9/65507
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
9Compounds containing elements of Groups 5 or 15 of the Periodic System
02Phosphorus compounds
547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
655having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms
65502the oxygen atom being part of a three-membered ring
65507condensed with carbocyclic rings or carbocyclic ring systems
Déposants
  • GILEAD SCIENCES, INC. [US/US]; 333 Lakeside Drive Foster City, CA 94404, US (AllExceptUS)
  • BOOJAMRA, Constantine, G. [US/US]; US (UsOnly)
  • CANNIZZARO, Carina, E. [AR/US]; US (UsOnly)
  • CHEN, James, M. [US/US]; US (UsOnly)
  • CHEN, Xiaowu [US/US]; US (UsOnly)
  • CHO, Aesop [US/US]; US (UsOnly)
  • CHONG, Lee, S. [US/US]; US (UsOnly)
  • DESAI, Manoj [US/US]; US (UsOnly)
  • FARDIS, Maria [US/US]; US (UsOnly)
  • GIBBS, Craig, S. [NZ/US]; US (UsOnly)
  • HIRSCHMANN, Ralph, F. [US/US]; US (UsOnly)
  • HUANG, Alan, X. [CN/US]; US (UsOnly)
  • JIN, Haolun [CA/US]; US (UsOnly)
  • KIM, Choung, U. [US/US]; US (UsOnly)
  • KIRSCHBERG, Thorsten, A. [DE/US]; US (UsOnly)
  • KRAWCZYK, Steven [US/US]; US (UsOnly)
  • LEE, Christopher, P. [US/US]; US (UsOnly)
  • LEE, William, A. [US/US]; US (UsOnly)
  • LIN, Kuei-Ying [US/US]; US (UsOnly)
  • MACKMAN, Richard, L. [GB/US]; US (UsOnly)
  • MARKEVITCH, David, Y. [RU/US]; US (UsOnly)
  • NELSON, Peter, H. [US/US]; US (UsOnly)
  • OARE, David, A. [US/US]; US (UsOnly)
  • PRASAD, Vidya, K. [SG/US]; US (UsOnly)
  • PYUN, Hyung-Jung [KR/US]; US (UsOnly)
  • RAY, Adrian, S. [US/US]; US (UsOnly)
  • SHERLOCK, Rosemarie [GB/US]; US (UsOnly)
  • SWAMINATHAN, Sundaramoorthi [IN/US]; US (UsOnly)
  • WATKINS, William, J. [GB/US]; US (UsOnly)
  • ZHANG, Jennifer, R. [US/US]; US (UsOnly)
  • ZHANG, Lijun [CN/US]; US (UsOnly)
Inventeurs
  • BOOJAMRA, Constantine, G.; US
  • CANNIZZARO, Carina, E.; US
  • CHEN, James, M.; US
  • CHEN, Xiaowu; US
  • CHO, Aesop; US
  • CHONG, Lee, S.; US
  • DESAI, Manoj; US
  • FARDIS, Maria; US
  • GIBBS, Craig, S.; US
  • HIRSCHMANN, Ralph, F.; US
  • HUANG, Alan, X.; US
  • JIN, Haolun; US
  • KIM, Choung, U.; US
  • KIRSCHBERG, Thorsten, A.; US
  • KRAWCZYK, Steven; US
  • LEE, Christopher, P.; US
  • LEE, William, A.; US
  • LIN, Kuei-Ying; US
  • MACKMAN, Richard, L.; US
  • MARKEVITCH, David, Y.; US
  • NELSON, Peter, H.; US
  • OARE, David, A.; US
  • PRASAD, Vidya, K.; US
  • PYUN, Hyung-Jung; US
  • RAY, Adrian, S.; US
  • SHERLOCK, Rosemarie; US
  • SWAMINATHAN, Sundaramoorthi; US
  • WATKINS, William, J.; US
  • ZHANG, Jennifer, R.; US
  • ZHANG, Lijun; US
Mandataires
  • BOSSE, Mark, L.; Gilead Sciences, Inc. 333 Lakeside Drive Foster City, CA 94404, US
Données relatives à la priorité
60/465,286 25.04.2003US
60/465,28725.04.2003US
60/465,28925.04.2003US
60/465,292 25.04.2003US
60/465,317 25.04.2003US
60/465,322 25.04.2003US
60/465,325 25.04.2003US
60/465,33225.04.2003US
60/465,33525.04.2003US
60/465,339 25.04.2003US
60/465,34225.04.2003US
60/465,34325.04.2003US
60/465,34725.04.2003US
60/465,355 25.04.2003US
60/465,373 25.04.2003US
60/465,377 25.04.2003US
60/465,380 25.04.2003US
60/465,39425.04.2003US
60/465,399 25.04.2003US
60/465,40025.04.2003US
60/465,40625.04.2003US
60/465,40825.04.2003US
60/465,415 25.04.2003US
60/465,419 25.04.2003US
60/465,420 25.04.2003US
60/465,42225.04.2003US
60/465,424 25.04.2003US
60/465,433 25.04.2003US
60/465,44925.04.2003US
60/465,45225.04.2003US
60/465,46325.04.2003US
60/465,46525.04.2003US
60/465,46725.04.2003US
60/465,46925.04.2003US
60/465,47125.04.2003US
60/465,47225.04.2003US
60/465,47325.04.2003US
60/465,475 25.04.2003US
60/465,47825.04.2003US
60/465,47925.04.2003US
60/465,48025.04.2003US
60/465,481 25.04.2003US
60/465,531 25.04.2003US
60/465,532 25.04.2003US
60/465,53625.04.2003US
60/465,53725.04.2003US
60/465,544 25.04.2003US
60/465,54525.04.2003US
60/465,54625.04.2003US
60/465,54725.04.2003US
60/465,54825.04.2003US
60/465,55025.04.2003US
60/465,55325.04.2003US
60/465,55425.04.2003US
60/465,55925.04.2003US
60/465,56025.04.2003US
60/465,56125.04.2003US
60/465,56725.04.2003US
60/465,56925.04.2003US
60/465,574 25.04.2003US
60/465,575 25.04.2003US
60/465,581 25.04.2003US
60/465,58425.04.2003US
60/465,58625.04.2003US
60/465,58725.04.2003US
60/465,58825.04.2003US
60/465,58925.04.2003US
60/465,59125.04.2003US
60/465,59325.04.2003US
60/465,59425.04.2003US
60/465,59825.04.2003US
60/465,60025.04.2003US
60/465,60125.04.2003US
60/465,60225.04.2003US
60/465,60325.04.2003US
60/465,60725.04.2003US
60/465,60825.04.2003US
60/465,61025.04.2003US
60/465,61425.04.2003US
60/465,62025.04.2003US
60/465,63025.04.2003US
60/465,63125.04.2003US
60/465,63225.04.2003US
60/465,63325.04.2003US
60/465,63425.04.2003US
60/465,63825.04.2003US
60/465,63925.04.2003US
60/465,64025.04.2003US
60/465,64125.04.2003US
60/465,64725.04.2003US
60/465,64925.04.2003US
60/465,658 25.04.2003US
60/465,66725.04.2003US
60/465,66825.04.2003US
60/465,68225.04.2003US
60/465,68325.04.2003US
60/465,68425.04.2003US
60/465,68725.04.2003US
60/465,689 25.04.2003US
60/465,69025.04.2003US
60/465,69525.04.2003US
60/465,69625.04.2003US
60/465,69825.04.2003US
60/465,71425.04.2003US
60/465,72025.04.2003US
60/465,72825.04.2003US
60/465,74225.04.2003US
60/465,74625.04.2003US
60/465,74925.04.2003US
60/465,751 25.04.2003US
60/465,756 25.04.2003US
60/465,75925.04.2003US
60/465,763 25.04.2003US
60/465,80525.04.2003US
60/465,82125.04.2003US
60/465,844 25.04.2003US
60/490,799 29.07.2003US
60/493,302 07.08.2003US
60/493,303 07.08.2003US
60/493,309 07.08.2003US
60/493,310 07.08.2003US
60/495,27315.08.2003US
60/495,274 15.08.2003US
60/495,27515.08.2003US
60/495,276 15.08.2003US
60/495,27715.08.2003US
60/495,27815.08.2003US
60/495,295 15.08.2003US
60/495,29715.08.2003US
60/495,29815.08.2003US
60/495,31715.08.2003US
60/495,33415.08.2003US
60/495,339 15.08.2003US
60/495,34115.08.2003US
60/495,34215.08.2003US
60/495,34315.08.2003US
60/495,34415.08.2003US
60/495,34515.08.2003US
60/495,347 15.08.2003US
60/495,34915.08.2003US
60/495,354 15.08.2003US
60/495,361 15.08.2003US
60/495,362 15.08.2003US
60/495,366 15.08.2003US
60/495,375 15.08.2003US
60/495,380 15.08.2003US
60/495,38215.08.2003US
60/495,38715.08.2003US
60/495,38815.08.2003US
60/495,389 15.08.2003US
60/495,39015.08.2003US
60/495,39115.08.2003US
60/495,392 15.08.2003US
60/495,393 15.08.2003US
60/495,398 15.08.2003US
60/495,414 15.08.2003US
60/495,416 15.08.2003US
60/495,417 15.08.2003US
60/495,425 15.08.2003US
60/495,426 15.08.2003US
60/495,427 15.08.2003US
60/495,43015.08.2003US
60/495,45315.08.2003US
60/495,455 15.08.2003US
60/495,456 15.08.2003US
60/495,460 15.08.2003US
60/495,471 15.08.2003US
60/495,472 15.08.2003US
60/495,48415.08.2003US
60/495,48515.08.2003US
60/495,48715.08.2003US
60/495,489 15.08.2003US
60/495,49015.08.2003US
60/495,49115.08.2003US
60/495,49215.08.2003US
60/495,524 15.08.2003US
60/495,52515.08.2003US
60/495,526 15.08.2003US
60/495,52715.08.2003US
60/495,529 15.08.2003US
60/495,530 15.08.2003US
60/495,531 15.08.2003US
60/495,532 15.08.2003US
60/495,533 15.08.2003US
60/495,534 15.08.2003US
60/495,537 15.08.2003US
60/495,53915.08.2003US
60/495,563 15.08.2003US
60/495,56415.08.2003US
60/495,565 15.08.2003US
60/495,59215.08.2003US
60/495,597 15.08.2003US
60/495,60015.08.2003US
60/495,60215.08.2003US
60/495,614 15.08.2003US
60/495,616 15.08.2003US
60/495,62915.08.2003US
60/495,63015.08.2003US
60/495,63115.08.2003US
60/495,63215.08.2003US
60/495,63315.08.2003US
60/495,64415.08.2003US
60/495,645 15.08.2003US
60/495,647 15.08.2003US
60/495,660 15.08.2003US
60/495,661 15.08.2003US
60/495,669 15.08.2003US
60/495,67115.08.2003US
60/495,679 15.08.2003US
60/495,680 15.08.2003US
60/495,681 15.08.2003US
60/495,68215.08.2003US
60/495,683 15.08.2003US
60/495,68415.08.2003US
60/495,68515.08.2003US
60/495,68615.08.2003US
60/495,68715.08.2003US
60/495,689 15.08.2003US
60/495,690 15.08.2003US
60/495,691 15.08.2003US
60/495,69615.08.2003US
60/495,736 15.08.2003US
60/495,748 15.08.2003US
60/495,749 15.08.2003US
60/495,751 15.08.2003US
60/495,753 15.08.2003US
60/495,754 15.08.2003US
60/495,75714.08.2003US
60/495,76015.08.2003US
60/495,762 15.08.2003US
60/495,76315.08.2003US
60/495,769 15.08.2003US
60/495,77215.08.2003US
60/495,784 15.08.2003US
60/495,789 15.08.2003US
60/495,80515.08.2003US
60/495,96415.08.2003US
60/510,245 10.10.2003US
60/513,530 24.10.2003US
60/513,531 24.10.2003US
60/513,561 24.10.2003US
60/513,562 24.10.2003US
60/513,563 24.10.2003US
60/513,564 24.10.2003US
60/513,579 24.10.2003US
60/513,58824.10.2003US
60/513,589 24.10.2003US
60/513,592 24.10.2003US
60/513,593 24.10.2003US
60/513,923 24.10.2003US
60/513,924 24.10.2003US
60/513,925 24.10.2003US
60/513,926 24.10.2003US
60/513,927 24.10.2003US
60/513,932 24.10.2003US
60/513,944 24.10.2003US
60/513,945 24.10.2003US
60/513,946 24.10.2003US
60/513,947 24.10.2003US
60/513,948 24.10.2003US
60/513,949 24.10.2003US
60/513,950 24.10.2003US
60/513,951 23.10.2003US
60/513,953 24.10.2003US
60/513,954 24.10.2003US
60/513,956 24.10.2003US
60/513,961 24.10.2003US
60/513,963 24.10.2003US
60/513,966 24.10.2003US
60/513,968 24.10.2003US
60/513,969 24.10.2003US
60/513,970 24.10.2003US
60/513,971 24.10.2003US
60/513,972 24.10.2003US
60/513,973 24.10.2003US
60/513,974 24.10.2003US
60/513,975 24.10.2003US
60/513,976 24.10.2003US
60/513,977 24.10.2003US
60/513,979 24.10.2003US
60/513,980 24.10.2003US
60/513,982 24.10.2003US
60/514,021 24.10.2003US
60/514,043 24.10.2003US
60/514,044 24.10.2003US
60/514,051 24.10.2003US
60/514,054 24.10.2003US
60/514,054 24.10.2003US
60/514,072 24.10.2003US
60/514,075 24.10.2003US
60/514,083 24.10.2003US
60/514,084 24.10.2003US
60/514,085 24.10.2003US
60/514,097 24.10.2003US
60/514,098 24.10.2003US
60/514,104 24.10.2003US
60/514,105 24.10.2003US
60/514,107 24.10.2003US
60/514,108 24.10.2003US
60/514,110 24.10.2003US
60/514,111 24.10.2003US
60/514,112 24.10.2003US
60/514,113 24.10.2003US
60/514,114 24.10.2003US
60/514,115 24.10.2003US
60/514,116 24.10.2003US
60/514,130 24.10.2003US
60/514,131 24.10.2003US
60/514,140 24.10.2003US
60/514,143 24.10.2003US
60/514,144 24.10.2003US
60/514,145 24.10.2003US
60/514,159 24.10.2003US
60/514,160 24.10.2003US
60/514,161 24.10.2003US
60/514,174 24.10.2003US
60/514,175 24.10.2003US
60/514,200 24.10.2003US
60/514,201 24.10.2003US
60/514,202 24.10.2003US
60/514,203 24.10.2003US
60/514,204 24.10.2003US
60/514,205 24.10.2003US
60/514,206 24.10.2003US
60/514,207 24.10.2003US
60/514,235 24.10.2003US
60/514,241 24.10.2003US
60/514,244 24.10.2003US
60/514,247 24.10.2003US
60/514,258 24.10.2003US
60/514,280 24.10.2003US
60/514,298 24.10.2003US
60/514,299 24.10.2003US
60/514,303 24.10.2003US
60/514,304 24.10.2003US
60/514,324 24.10.2003US
60/514,325 24.10.2003US
60/514,326 24.10.2003US
60/514,330 24.10.2003US
60/514,334 24.10.2003US
60/514,345 24.10.2003US
60/514,346 24.10.2003US
60/514,359 24.10.2003US
60/514,360 24.10.2003US
60/514,368 24.10.2003US
60/514,369 24.10.2003US
60/514,393 24.10.2003US
60/514,394 24.10.2003US
60/514,424 24.10.2003US
60/514,439 24.10.2003US
60/514,450 24.10.2003US
60/514,452 24.10.2003US
60/514,453 24.10.2003US
60/514,461 24.10.2003US
60/514,462 24.10.2003US
60/514,464 24.10.2003US
60/514,465 24.10.2003US
60/514,466 24.10.2003US
60/514,481 24.10.2003US
60/514,522 24.10.2003US
60/515,266 29.10.2003US
60/519,476 12.11.2003US
60/524,340 20.11.2003US
60/531,932 22.12.2003US
60/531,940 22.12.2003US
60/531,960 22.12.2003US
60/532,160 22.12.2003US
60/532,183 22.12.2003US
60/532,184 22.12.2003US
60/532,230 22.12.2003US
60/532,257 22.12.2003US
60/532,273 22.12.2003US
60/532,274 22.12.2003US
60/532,415 23.12.2003US
60/532,587 23.12.2003US
60/532,591 23.12.2003US
60/532,682 23.12.2003US
60/532,683 23.12.2003US
60/536,003 12.01.2004US
60/536,004 12.01.2004US
60/536,005 12.01.2004US
60/536,006 12.01.2004US
60/536,007 12.01.2004US
60/536,009 12.01.2004US
60/536,027 12.01.2004US
60/536,054 12.01.2004US
60/536,179 12.01.2004US
60/536,180 12.01.2004US
Langue de publication anglais (EN)
Langue de dépôt anglais (EN)
États désignés
Titre
(EN) THERAPEUTIC PHOSPHONATE COMPOUNDS
(FR) COMPOSES DE PHOSPHONATE THERAPEUTIQUES
Abrégé
(EN)
The invention is related to phosphorus substituted therapeutic agents, compositions containing such phosphorus substituted agents, and therapeutic methods that include the administration of such phosphorus substituted agents, as well as to processes and intermediates useful for preparing such agents.
(FR)
La présente invention a trait à des agents thérapeutiques substitués de phosphore, des compositions contenant de tels agents substitués de phosphore, et des procédés thérapeutiques comprenant l'administration de tels agents substitués de phosphore, ainsi que des procédés et des intermédiaires utiles pour la préparation de tels agents.
Également publié en tant que
US11258621
Dernières données bibliographiques dont dispose le Bureau international