処理中

しばらくお待ちください...

設定

設定

出願の表示

1. WO2005034953 - 血管新生抑制薬

公開番号 WO/2005/034953
公開日 21.04.2005
国際出願番号 PCT/JP2004/014956
国際出願日 08.10.2004
IPC
A61K 31/444 2006.01
A生活必需品
61医学または獣医学;衛生学
K医薬用,歯科用又は化粧用製剤
31有機活性成分を含有する医薬品製剤
33複素環式化合物
395環異種原子として窒素を持つもの,例.グアネチジン,リファマイシン
435環異種原子として1個の窒素のみを有する6員環を持つもの,例.炭素環系と縮合したもの
44非縮合ピリジン;その水素添加誘導体
4427さらに複素環系を含有するもの
444環異種原子として窒素を有する6員環を含むもの,例.アムリノン
C07D 401/14 2006.01
C化学;冶金
07有機化学
D複素環式化合物(高分子化合物C08)
401異項原子として窒素原子のみをもつ2個以上の複素環を含有し,そのうち少なくても1個が1個の窒素原子のみをもつ6員環である複素環式化合物
143個以上の複素環を含有するもの
CPC
A61K 31/444
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
435having six-membered rings with one nitrogen as the only ring hetero atom
44Non condensed pyridines; Hydrogenated derivatives thereof
4427containing further heterocyclic ring systems
444containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
A61K 31/4468
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
435having six-membered rings with one nitrogen as the only ring hetero atom
44Non condensed pyridines; Hydrogenated derivatives thereof
445Non condensed piperidines, e.g. piperocaine
4468having a nitrogen directly attached in position 4, e.g. clebopride, fentanyl
A61K 31/4545
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
435having six-membered rings with one nitrogen as the only ring hetero atom
44Non condensed pyridines; Hydrogenated derivatives thereof
445Non condensed piperidines, e.g. piperocaine
4523containing further heterocyclic ring systems
4545containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
A61P 27/02
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
27Drugs for disorders of the senses
02Ophthalmic agents
A61P 27/06
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
27Drugs for disorders of the senses
02Ophthalmic agents
06Antiglaucoma agents or miotics
A61P 3/10
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
3Drugs for disorders of the metabolism
08for glucose homeostasis
10for hyperglycaemia, e.g. antidiabetics
出願人
  • 興和株式会社 KOWA CO., LTD. [JP]/[JP] (AllExceptUS)
  • 土肥 武 DOI, Takeshi [JP]/[JP] (UsOnly)
  • 田村 正宏 TAMURA, Masahiro [JP]/[JP] (UsOnly)
発明者
  • 土肥 武 DOI, Takeshi
  • 田村 正宏 TAMURA, Masahiro
代理人
  • 特許業務法人アルガ特許事務所 THE PATENT CORPORATE BODY ARUGA PATENT OFFICE
優先権情報
60/510,01210.10.2003US
公開言語 (言語コード) 日本語 (JA)
出願言語 (言語コード) 日本語 (JA)
指定国 (国コード)
発明の名称
(EN) ANGIOGENESIS INHIBITOR
(FR) INHIBITEUR D'ANGIOGENESE
(JA) 血管新生抑制薬
要約
(EN)
A preventive/therapeutic agent for diseases attributable to angiogenesis which contains as an active ingredient a cyclic amine compound represented by the general formula (1): (Chemical formula 1) (1) (wherein R1, R2, and R3 each independently represents hydrogen, halogeno, hydroxy, alkyl, halogenoalkyl, alkoxy, alkylthio, carboxy, alkoxycarbonyl, or alkanoyl; W1 and W2 each independently represents nitrogen or CH; X represents oxygen, NR4, CONR4, or NR4CO; R4's each represents hydrogen, alkyl, alkenyl, alkynyl, (un)substituted aryl, (un)substituted heteroaryl, (un)substituted aralkyl, or (un)substituted heteroaralkyl; and l, m, and n each is 0 or 1), a salt of the compound, or a solvate of either.
(FR)
Agent préventif / thérapeutique destiné à combattre les maladies attribuées à l'angiogenèse, qui contient en tant qu'ingrédient actif un composé d'amine cyclique représentée par la formule générale (1): (formule chimique 1) (1) (dans laquelle R1, R2, et R3 représente chacun indépendamment hydrogène, halogéno, hydroxy, alkyl, halogéno-alkyl, alcoxy, alkylthio, carboxy, alcoxycarbonyl, ou alcanoyl; W1 et W2 représente chacun indépendamment azote ou CH; X représente oxygène, NR4, CONR4 ou NR4CO; R4 représente chacun hydrogène, alkyle, alcényle, alkynyl, aryl (non)substitué, hétéroaryle (non)substitué, aralalkyle (non)substitué ou hétéro- aralalkyle (non)substitué; et l, m, et n sont chacun ou or 1), un sel du composé ou un solvat du composé ou du sel.
(JA)
not available
他の公開
US2007043078
国際事務局に記録されている最新の書誌情報