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1. WO2012009226 - IMIDAZOLONES SUBSTITUÉS, COMPOSITIONS CONTENANT CES COMPOSÉS, ET PROCÉDÉS D'UTILISATION

Numéro de publication WO/2012/009226
Date de publication 19.01.2012
N° de la demande internationale PCT/US2011/043369
Date du dépôt international 08.07.2011
CIB
A01N 43/50 2006.01
ANÉCESSITÉS COURANTES DE LA VIE
01AGRICULTURE; SYLVICULTURE; ÉLEVAGE; CHASSE; PIÉGEAGE; PÊCHE
NCONSERVATION DE CORPS HUMAINS OU ANIMAUX OU DE VÉGÉTAUX, OU DE PARTIES DE CEUX-CI; BIOCIDES, p.ex. EN TANT QUE DÉSINFECTANTS, PESTICIDES OU HERBICIDES; PRODUITS REPOUSSANT OU ATTIRANT LES ANIMAUX NUISIBLES; RÉGULATEURS DE CROISSANCE DES VÉGÉTAUX
43Biocides, produits repoussant ou attirant les animaux nuisibles, ou régulateurs de croissance des végétaux, contenant des composés hétérocycliques
48comportant des cycles avec deux atomes d'azote comme uniques hétéro-atomes du cycle
50Diazoles-1,3; Diazoles-1,3 hydrogénés
CPC
A61K 31/4166
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
41having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
41641,3-Diazoles
4166having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
A61K 31/4178
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
41having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
41641,3-Diazoles
4178not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
C07D 233/36
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
233Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
04having one double bond between ring members or between a ring member and a non-ring member
28with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
30Oxygen or sulfur atoms
32One oxygen atom
36with hydrocarbon radicals, substituted by nitrogen atoms, attached to ring nitrogen atoms
C07D 233/70
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
233Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
54having two double bonds between ring members or between ring members and non-ring members
66with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
70One oxygen atom
C07D 403/12
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
403Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
02containing two hetero rings
12linked by a chain containing hetero atoms as chain links
Déposants
  • MERCK SHARP & DOHME CORP. [US/US]; 126 East Lincoln Avenue Rahway, New Jersey 07065-0907, US (AllExceptUS)
  • DEMONG, Duane [US/US]; US (NZ, US)
  • MILLER, Michael, W. [US/US]; US (NZ, US)
  • DAI, Xing [CN/US]; US (NZ, US)
  • STAMFORD, Andrew [AU/US]; US (NZ, US)
Inventeurs
  • DEMONG, Duane; US
  • MILLER, Michael, W.; US
  • DAI, Xing; US
  • STAMFORD, Andrew; US
Représentant commun
  • MERCK SHARP & DOHME CORP.; 126 East Lincoln Avenue Rahway, NJ 07065-0907, US
Données relatives à la priorité
61/363,81213.07.2010US
Langue de publication anglais (EN)
Langue de dépôt anglais (EN)
États désignés
Titre
(EN) SUBSTITUTED IMIDAZOLONES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE
(FR) IMIDAZOLONES SUBSTITUÉS, COMPOSITIONS CONTENANT CES COMPOSÉS, ET PROCÉDÉS D'UTILISATION
Abrégé
(EN)
The present invention relates to compounds of the general structure shown in Formula (A): (A): and includes pharmaceutically acceptable salts, solvates, esters, prodrugs, tautomers, and isomers of said compounds. Pharmaceutical compositions and methods of treatment are also included.
(FR)
La présente invention concerne des composés de structure générale montrée dans la formule (A) : (A) : qui comprennent des sels pharmaceutiqument acceptables, des solvates, des esters, des promédicaments, des tautomères et des isomères desdits composés. L'invention porte en outre sur des compositions pharmaceutiques et des procédés de traitement.
Également publié en tant que
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