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1. WO2022010175 - PHARMACEUTICAL COMPOSITIONS COMPRISING A DIAMINOPYRIMIDINE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF AND PROCESSES FOR PREPARING THE SAME

Publication Number WO/2022/010175
Publication Date 13.01.2022
International Application No. PCT/KR2021/008327
International Filing Date 01.07.2021
IPC
A61K 9/20 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
9Medicinal preparations characterised by special physical form
20Pills, lozenges or tablets
A61K 47/12 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
47Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
08containing oxygen
12Carboxylic acids; Salts or anhydrides thereof
A61K 31/506 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
495having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
506not condensed and containing further heterocyclic rings
A61P 1/00 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
1Drugs for disorders of the alimentary tract or the digestive system
Applicants
  • YUHAN CORPORATION [KR]/[KR]
Inventors
  • PARK, Dong-Min
  • KIM, Su-Hyeon
  • CHEON, Eun-Pa
  • HA, Tae-Lin
  • YANG, Jun-Mo
  • PARK, Yoong-Sik
Agents
  • OH, Kook-Jin
Priority Data
10-2020-008459509.07.2020KR
Publication Language English (en)
Filing Language English (EN)
Designated States
Title
(EN) PHARMACEUTICAL COMPOSITIONS COMPRISING A DIAMINOPYRIMIDINE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF AND PROCESSES FOR PREPARING THE SAME
(FR) COMPOSITIONS PHARMACEUTIQUES COMPRENANT UN DÉRIVÉ DE DIAMINOPYRIMIDINE OU UN SEL PHARMACEUTIQUEMENT ACCEPTABLE DE CELUI-CI ET LEURS PROCÉDÉS DE PRÉPARATION
Abstract
(EN) The present invention provides a pharmaceutical composition comprising (S)-N-(1-(2-((4-amino-3-nitrophenyl)amino)-6-propylpyrimidin-4-yl)pyrrolidin-3-yl)acetamide or a pharmaceutically acceptable salt thereof having an activity as a 5-HT4 receptor agonist and an acidifying agent; and a process for preparing the same.
(FR) La présente invention concerne une composition pharmaceutique comprenant (S)-N-(1-(2-((4-amino-3-nitrophényle)amino)-6-propylpyrimidine-4-yl) pyrrolidine-3-yl)acétamide ou un sel pharmaceutiquement acceptable de celui-ci ayant une activité en tant qu'agoniste du récepteur 5-HT4 et un agent acidifiant ; et son procédé de préparation.
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