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1. WO2022002780 - TETRAZOLE DERIVATIVES AS TRPA1 INHIBITORS

Publication Number WO/2022/002780
Publication Date 06.01.2022
International Application No. PCT/EP2021/067467
International Filing Date 25.06.2021
IPC
A61K 31/5365 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
535having six-membered rings with at least one nitrogen and at least one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
5365ortho- or peri-condensed with heterocyclic ring systems
A61K 31/519 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
495having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
519ortho- or peri-condensed with heterocyclic rings
A61K 31/54 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
54having six-membered rings with at least one nitrogen and at least one sulfur as the ring hetero atoms, e.g. sulthiame
Applicants
  • BOEHRINGER INGELHEIM INTERNATIONAL GMBH [DE]/[DE]
Inventors
  • FLECK, Martin, Thomas
  • BINDER, Florian, Paul, Christian
  • WILLWACHER, Jens
Agents
  • SIMON, Elke, Anna, Maria
  • SEITZ, Dr. Jürgen
Priority Data
20182987.629.06.2020EP
Publication Language English (en)
Filing Language English (EN)
Designated States
Title
(EN) TETRAZOLE DERIVATIVES AS TRPA1 INHIBITORS
(FR) DÉRIVÉS DE TÉTRAZOLE UTILES EN TANT QU'INHIBITEURS DE TRPA1
Abstract
(EN) The present disclosure provides certain tetrazole derivatives that are inhibitors of transient receptor potential ankyrin 1 (TRPA1), and are therefore useful for the treatment of diseases treatable by inhibition of TRPA1. Also provided are pharmaceutical compositions containing the same, and processes for preparing said compounds.
(FR) La présente invention concerne certains dérivés de tétrazole qui sont des inhibiteurs de l'ankyrine à potentiel récepteur transitoire 1 (TRPA1) et sont par conséquent utiles pour le traitement de maladies pouvant être traitées par inhibition de TRPA1. L'invention concerne également des compositions pharmaceutiques les contenant et des procédés de préparation desdits composés.
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