Processing

Please wait...

Settings

Settings

Goto Application

1. WO2021059160 - PROCESS FOR PREPARING 5-(FLUORO-4-IMINO-3-METHYL)-1-TOSYL-3,4 DIHYDROPYRIMIDINE -(1H)-ONE

Publication Number WO/2021/059160
Publication Date 01.04.2021
International Application No. PCT/IB2020/058893
International Filing Date 23.09.2020
IPC
C07D 239/47 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
239Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
02not condensed with other rings
24having three or more double bonds between ring members or between ring members and non-ring members
28with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
46Two or more oxygen, sulfur or nitrogen atoms
47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
A01N 43/54 2006.01
AHUMAN NECESSITIES
01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
48having rings with two nitrogen atoms as the only ring hetero atoms
541,3-Diazines; Hydrogenated 1,3-diazines
A01N 43/56 2006.01
AHUMAN NECESSITIES
01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
48having rings with two nitrogen atoms as the only ring hetero atoms
561,2-Diazoles; Hydrogenated 1,2-diazoles
A01N 43/653 2006.01
AHUMAN NECESSITIES
01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
64having rings with three nitrogen atoms as the only ring hetero atoms
647Triazoles; Hydrogenated triazoles
6531,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
CPC
A01N 43/54
AHUMAN NECESSITIES
01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES
43Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
48having rings with two nitrogen atoms as the only ring hetero atoms
541,3-Diazines; Hydrogenated 1,3-diazines
C07D 239/47
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
239Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
02not condensed with other rings
24having three or more double bonds between ring members or between ring members and non-ring members
28with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
46Two or more oxygen, sulfur or nitrogen atoms
47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
Applicants
  • ADAMA MAKHTESHIM LTD. [IL]/[IL]
  • SUEZ, Gal [IL]/[IL] (US)
  • ALASIBI, Samaa [IL]/[IL] (US)
  • MINES, Yaakov [IL]/[IL] (US)
Inventors
  • SUEZ, Gal
  • ALASIBI, Samaa
  • MINES, Yaakov
Priority Data
62/904,48223.09.2019US
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) PROCESS FOR PREPARING 5-(FLUORO-4-IMINO-3-METHYL)-1-TOSYL-3,4 DIHYDROPYRIMIDINE -(1H)-ONE
(FR) PROCÉDÉ DE PRÉPARATION DE 5-(FLUORO-4-IMINO-3-MÉTHYL)-1-TOSYL-3,4-DIHYDROPYRIMIDINE-(1H)-ONE
Abstract
(EN)
The present invention provides a process for preparing a compound having the formula (I): wherein R is alkyl or alkylaryl; each of X1, X2, X3, X4 and X5 is, independently, H, alkyl, alkenyl, alkynyl, alkoxy, haloalkyl, haloalkoxy, alkylthio, haloalkylthio, amino, alkylamino, dialkylamino, alkoxycarbonyl, alkyl carbonyl, hydroxyalkyl, ester, acid, halogen, -SH, -OH, -NH2, -NO2, -CN or CF3; Y is O or S; and and Z is a halogen.
(FR)
La présente invention concerne un procédé de préparation d'un composé de formule (I) : dans laquelle R représente un alkyle ou un alkylaryle; chacun de X1, X2, X3, X4 et X5 représente indépendamment H, un alkyle, un alcényle, un alcynyle, un alcoxy, un halogénoalkyle, un halogénoalcoxy, un alkylthio, un halogénoalkylthio, un amino, un alkylamino, un dialkylamino, un alcoxycarbonyle, un alkylcarbonyle, un hydroxyalkyle, un ester, un acide, un halogène, -SH, -OH, -NH2, -NO2, -CN ou CF3; Y représente O ou S; et Z représente un halogène.
Latest bibliographic data on file with the International Bureau