Processing

Please wait...

Settings

Settings

Goto Application

1. WO2021055589 - HETEROARYL PLASMA KALLIKREIN INHIBITORS

Publication Number WO/2021/055589
Publication Date 25.03.2021
International Application No. PCT/US2020/051249
International Filing Date 17.09.2020
IPC
A61P 29/02 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
29Non-central analgesic, antipyretic or antiinflammatory agents, e.g antirheumatic agents; Non-steroidal antiinflammatory drugs (NSAIDs)
02without antiinflammatory effect
A61K 31/495 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
495having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
C07D 519/00 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
519Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/ or C07D455/257
Applicants
  • TAKEDA PHARMACEUTICAL COMPANY LIMITED [JP]/[JP]
Inventors
  • PAPAIOANNOU, Nikolaos
  • TRAVINS, Jeremy Mark
  • FINK, Sarah Jocelyn
  • ELLARD, John Mark
  • RAE, Alastair
Agents
  • REARICK, John P.
  • ADAMS, Melissa M.
  • ADATO, Ronen
  • AUGST, Alexander
  • BUTEAU, Kristen C.
  • BYCHOWSKI, Meaghan E.
  • D'AMATO, Erica M.
  • DAUKSS, Dana M.
  • FLYNN, Peter A.
  • HAULBROOK, William R.
  • JARRELL, Brenda Herschbach
  • JUDA, Cristin E.
  • LI, Xiaodong
  • LYON, Charles E.
  • MA, Longle
  • MEDINA, Rolando
  • MONROE, Margo R.
  • PACE, Nicholas J.
  • POLIO, Samuel R.
  • REESE, Brian E.
  • SCHMITT, Michael
  • SCHONEWALD, Stephanie L.
  • SHINALL, Michael A.
  • SHORE, David E.
  • SMITH, Maria C.
  • SUBRAMANIAN, Sowmya
  • SUH, Su Kyung
  • TSE, Janet M.
  • VETTER, Michael L.
  • VRABLIK, Tracy L.
  • ZHANG, Jialan
Priority Data
62/902,33318.09.2019US
Publication Language English (en)
Filing Language English (EN)
Designated States
Title
(EN) HETEROARYL PLASMA KALLIKREIN INHIBITORS
(FR) INHIBITEURS HÉTÉROARYLES DE LA KALLICRÉINE PLASMATIQUE
Abstract
(EN) The present invention provides compounds and compositions thereof which are useful as inhibitors of plasma kallikrein and which exhibit desirable characteristics for the same.
(FR) La présente invention concerne des composés et des compositions de ceux-ci qui sont utiles en tant qu'inhibiteurs de la kallicréine plasmatique et qui présentent des caractéristiques souhaitables pour ceux-ci.
Related patent documents
EP2020781702This application is not viewable in PATENTSCOPE because the national phase entry has not been published yet or the national entry is issued from a country that does not share data with WIPO or there is a formatting issue or an unavailability of the application.
Latest bibliographic data on file with the International Bureau