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1. WO2020210785 - D3 RECEPTOR AGONIST COMPOUNDS; METHODS OF PREPARATION; INTERMEDIATES THEREOF; AND METHODS OF USE THEREOF

Publication Number WO/2020/210785
Publication Date 15.10.2020
International Application No. PCT/US2020/027903
International Filing Date 13.04.2020
IPC
C07D 413/14 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
413Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
14containing three or more hetero rings
A61K 31/5377 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
535having six-membered rings with at least one nitrogen and at least one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
53751,4-Oxazines, e.g. morpholine
5377not condensed and containing further heterocyclic rings, e.g. timolol
A61P 25/00 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25Drugs for disorders of the nervous system
CPC
C07D 413/14
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
413Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
14containing three or more hetero rings
Applicants
  • THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES [US]/[US]
Inventors
  • HAUCK NEWMAN, Amy
  • BONIFAZI, Alessandro
  • BATTITI, Francisco, Oscar
  • CEMAJ, Sophie, L.
Agents
  • PELLETIER, Roberta, L.
Priority Data
62/833,02312.04.2019US
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) D3 RECEPTOR AGONIST COMPOUNDS; METHODS OF PREPARATION; INTERMEDIATES THEREOF; AND METHODS OF USE THEREOF
(FR) COMPOSÉS AGONISTES DU RÉCEPTEUR D3; PROCÉDÉS DE PRÉPARATION; INTERMÉDIAIRES DE CEUX-CI; ET LEURS PROCÉDÉS D'UTILISATION
Abstract
(EN)
Disclosed herein are novel compounds including dopamine D3 receptor agonists, compositions thereof, methods of use thereof, and processes of synthesizing the same. Further disclosed are D3R selective agonist compounds, specifically bitopic ligands comprising chirality.
(FR)
L'invention concerne de nouveaux composés comprenant des agonistes du récepteur D3 de la dopamine, des compositions de ceux-ci, des procédés d'utilisation de ceux-ci, et des procédés de synthèse de ceux-ci. L'invention concerne en outre des composés agonistes sélectifs de D3R, en particulier des ligands bitopiques comprenant une chiralité.
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