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1. WO2020204024 - THYMINE NUCLEOBASE-BASED TRIAZOLOPYRIMIDINES AND PRODUCTION METHOD THEREFOR

Publication Number WO/2020/204024
Publication Date 08.10.2020
International Application No. PCT/JP2020/014810
International Filing Date 31.03.2020
IPC
A61P 35/00 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
35Antineoplastic agents
C07D 487/04 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
487Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/-C07D477/183
02in which the condensed system contains two hetero rings
04Ortho-condensed systems
A61K 31/519 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
495having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
519ortho- or peri-condensed with heterocyclic rings
Applicants
  • テラ・ストーン株式会社 TERA STONE CO., LTD [JP]/[JP]
Inventors
  • 永松 朝文 NAGAMATSU, Tomohisa
Agents
  • 森本 敏明 MORIMOTO, Toshiaki
Priority Data
2019-07152503.04.2019JP
Publication Language Japanese (JA)
Filing Language Japanese (JA)
Designated States
Title
(EN) THYMINE NUCLEOBASE-BASED TRIAZOLOPYRIMIDINES AND PRODUCTION METHOD THEREFOR
(FR) TRIAZOLOPYRIMIDINES À BASE DE NUCLÉOBASE DE TYPE THYMINE ET PROCÉDÉ DE PRODUCTION ASSOCIÉ
(JA) チミン核酸塩基をベースとするトリアゾロピリミジン類及びその製造方法
Abstract
(EN)
Provided are: novel triazolopyrimidines that can be induced from the nucleobase thymine; a production method for the triazolopyrimidines; and various physiologically active substances, particularly an antitumor agent, obtained by the method. These triazolopyrimidine compounds are represented by formulas (I)-(VIII) (in the formulas, R represents a hydrogen atom, an alkyl group, or an aryl group). This production method produces the triazolopyrimidine compounds.
(FR)
L'invention concerne : de nouvelles triazolopyrimidines qui peuvent être induites à partir de la nucléobase de type thymine ; un procédé de production des triazolopyrimidines ; et diverses substances physiologiquement actives, en particulier un agent antitumoral, obtenues par le procédé. Ces composés de triazolopyrimidine sont représentés par les formules (I)-(VIII) (dans les formules, R représente un atome d'hydrogène, un groupe alkyle ou un groupe aryle). Ce procédé de production produit les composés de triazolopyrimidine.
(JA)
核酸塩基のチミンから誘導できる新規トリアゾロピリミジン類及びその製造方法、該方法よって得られる種々の生理活性物質、特に抗腫瘍剤を提供する。下記式(I)から(VIII)で表されるトリアゾロピリミジン類化合物(式中、Rは水素原子、アルキル基又はアリール基を示す)及び該化合物の製造方法。
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