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1. WO2020112542 - COMBINATION COMPOSITIONS COMPRISING A BETA-LACTAMASE INHIBITOR AND USES THEREOF

Publication Number WO/2020/112542
Publication Date 04.06.2020
International Application No. PCT/US2019/062798
International Filing Date 22.11.2019
IPC
A61K 8/37 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
8Cosmetics or similar toilet preparations
18characterised by the composition
30containing organic compounds
33containing oxygen
37Esters of carboxylic acids
A61K 31/69 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
69Boron compounds
C07C 29/52 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
29Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
48by oxidation reactions with formation of hydroxy groups
50with molecular oxygen only
52in the presence of mineral boron compounds with, when necessary, hydrolysis of the intermediate formed
C07C 63/06 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
63Compounds having carboxyl groups bound to carbon atoms of six-membered aromatic rings
04Monocyclic monocarboxylic acids
06Benzoic acid
CPC
A61K 31/69
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
69Boron compounds
C07C 29/52
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
29Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
48by oxidation reactions with formation of hydroxy groups
50with molecular oxygen only
52in the presence of mineral boron compounds with, when necessary, hydrolysis of the intermediate formed
C07C 63/06
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
63Compounds having carboxyl groups bound to a carbon atoms of six-membered aromatic rings
04Monocyclic monocarboxylic acids
06Benzoic acid
Applicants
  • VENATORX PHARMACEUTICALS, INC. [US]/[US]
Inventors
  • BURNS, Christopher J.
  • DAIGLE, Denis
  • HAMRICK, Jodie
  • PEVEAR, Daniel C.
  • TROUT, Robert E. Lee
  • XERRI, Luigi
  • HENKEL, Timothy
  • MYERS, Cullen L.
  • CONDON, Stephen M.
  • DRAGER, Anthony
  • ROSEN, Lawrence
Agents
  • HARDT, Ingo H.
Priority Data
62/773,06329.11.2018US
62/777,64310.12.2018US
62/796,52424.01.2019US
62/828,35402.04.2019US
62/832,11810.04.2019US
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) COMBINATION COMPOSITIONS COMPRISING A BETA-LACTAMASE INHIBITOR AND USES THEREOF
(FR) COMPOSITIONS MIXTES COMPRENANT UN INHIBITEUR DE BÊTA-LACTAMASE ET LEURS UTILISATIONS
Abstract
(EN)
The present invention relates to pharmaceutical compositions containing boron-containing compounds and their use as inhibitors of beta-lactamase enzymes and as antibacterial agents in combination with a beta-lactam antibiotic.
(FR)
La présente invention concerne des compositions pharmaceutiques contenant des composés contenant du bore et leur utilisation en tant qu'inhibiteurs d'enzymes bêta-lactamase et en tant qu'agents antibactériens en combinaison avec un antibiotique bêta-lactame.
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