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1. WO2020090585 - (HETERO)ARYLIMIDAZOLE COMPOUND AND HARMFUL ORGANISM CONTROL AGENT

Publication Number WO/2020/090585
Publication Date 07.05.2020
International Application No. PCT/JP2019/041540
International Filing Date 23.10.2019
IPC
C07D 233/64 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
233Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
54having two double bonds between ring members or between ring members and non-ring members
64with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
A01N 43/50 2006.01
AHUMAN NECESSITIES
01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
48having rings with two nitrogen atoms as the only ring hetero atoms
501,3-Diazoles; Hydrogenated 1,3-diazoles
A01P 7/02 2006.01
AHUMAN NECESSITIES
01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
PBIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
7Arthropodicides
02Acaricides
A01P 7/04 2006.01
AHUMAN NECESSITIES
01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
PBIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
7Arthropodicides
04Insecticides
A61K 31/4164 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
41having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole
41641,3-Diazoles
A61K 31/4439 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
435having six-membered rings with one nitrogen as the only ring hetero atom
44Non-condensed pyridines; Hydrogenated derivatives thereof
4427containing further heterocyclic ring systems
4439containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
Applicants
  • 日本曹達株式会社 NIPPON SODA CO., LTD. [JP]/[JP]
Inventors
  • 阪西 慶太 SAKANISHI, Keita
  • 崎山 訓史 SAKIYAMA, Norifumi
  • 青山 光 AOYAMA, Hikaru
  • 松井 麻記 MATSUI, Maki
  • 岩佐 孝男 IWASA, Takao
  • 小林 朝巳 KOBAYASHI, Tomomi
  • 牛島 大佑 USHIJIMA, Daisuke
  • 東 慶太 AZUMA, Keita
  • 住野 正憲 SUMINO, Masanori
  • 芦刈 康彦 ASHIKARI, Yasuhiko
  • 柴山 耕太郎 SHIBAYAMA, Kotaro
  • 田口 莉帆 TAGUCHI, Riho
Agents
  • 廣田 雅紀 HIROTA, Masanori
Priority Data
2018-20299829.10.2018JP
Publication Language Japanese (JA)
Filing Language Japanese (JA)
Designated States
Title
(EN) (HETERO)ARYLIMIDAZOLE COMPOUND AND HARMFUL ORGANISM CONTROL AGENT
(FR) COMPOSÉ (HÉTÉRO)ARYLIMIDAZOLE ET AGENT DE LUTTE CONTRE LES ORGANISMES NUISIBLES
(JA) (ヘテロ)アリールイミダゾール化合物および有害生物防除剤
Abstract
(EN)
The present invention addresses the problem of providing a (hetero)arylimidazole compound which has an excellent harmful organism controlling activity, particularly an excellent insecticidal activity and/or an excellent acaricidal activity, also has excellent safety, and can be synthesized industrially advantageously. The (hetero)arylimidazole compound according to the present invention is a compound represented by formula (I), or an N-oxide compound, a stereoisomer, a tautomer or a hydrate of the compound, or a salt of the compound, the N-oxide compound, the stereoisomer, the tautomer or the hydrate. In formula (I), B1 represents a nitrogen atom or CH; X represents a substituted or unsubstituted C3-8 cycloalkyl group; R1 represents a substituted or unsubstituted C1-6 alkylthio group or a substituted or unsubstituted C1-6 alkylsulfonyl group; R2 represents a substituted or unsubstituted C1-6 alkyl group; and R represents a substituted or unsubstituted C2-6 alkenyl group.
(FR)
Le problème décrit par la présente invention concerne la fourniture d'un composé (hétéro)arylimidazole qui a une excellente activité de lutte contre les organismes nuisibles, en particulier, une excellente activité insecticide et/ou une excellente activité acaricide, ainsi qu'une sécurité élevée, et peut être synthétisé de manière avantageuse sur le plan industriel. Le composé (hétéro)arylimidazole selon la présente invention est un composé de formule (I), ou un composé N-oxyde, un stéréoisomère, un tautomère ou un hydrate du composé, ou un sel du composé, du composé N-oxyde, du stéréoisomère, du tautomère ou de l'hydrate. Dans la formule (I), B1 représente un atome d'azote ou CH ; X représente un groupe cycloalkyle en C3-8 substitué ou non substitué ; R1 représente un groupe alkylthio en C1-6 substitué ou non substitué ou un groupe alkylsulfonyle en C1-6 substitué ou non substitué ; R2 représente un groupe alkyle en C1-6 substitué ou non substitué ; et R représente un groupe alcényle en C2-6 substitué ou non substitué.
(JA)
本発明の課題は、有害生物防除活性、その中でも特に殺虫活性および/または殺ダニ活性に優れ、安全性に優れ、かつ工業的に有利に合成できる(ヘテロ)アリールイミダゾール化合物を提供することである。 本発明の(ヘテロ)アリールイミダゾール化合物は、式(I)で表される化合物、そのN-オキサイド化合物、立体異性体、互変異性体、水和物またはそれらの塩である。 式(I)中、 B1は、窒素原子、またはCHであり、Xは、置換若しくは無置換のC3~8シクロアルキル基であり、R1は、置換若しくは無置換のC1~6アルキルチオ基、または置換若しくは無置換のC1~6アルキルスルホニル基であり、R2は、置換若しくは無置換のC1~6アルキル基であり、且つRは、置換若しくは無置換のC2~6アルケニル基である。
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