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1. WO2020070049 - PESTICIDALLY ACTIVE BENZENE- AND AZINE-AMIDE COMPOUNDS

Note: Text based on automatic Optical Character Recognition processes. Please use the PDF version for legal matters

[ EN ]

CLAIMS

1. A compound of the formula I


wherein:

Q is


Ai, A2, A3 and A4 are independently CRs or N, provided not more than three of A1, A2, A3 and A4 are N; R1 is hydrogen, Ci-C6alkyl, Ci-C6cyanoalkyl, aminocarbonylCi-Cealkyl, hydroxycarbonylC-i-Cealkyl, C1-Cenitroalkyl, trimethylsilaneCi-Cealkyl, Ci-C6haloalkyl, C2-C6alkenyl, C2-C6haloalkenyl, C2-C6alkynyl, C2-C6haloalkynyl; C3-C4cycloalkylCi-C2alkyl- wherein the C3-C4cycloalkyl is optionally substituted with 1 or 2 halo atoms; oxetan-3-yl-CH2-; or benzyl optionally substituted with halo or Ci-C6haloalkyl;

R2 is phenyl, pyridine, pyrimidine, pyrazine or pyridazine, wherein the phenyl, pyridine, pyrimidine, pyrazine or pyridazine is optionally substituted with one to three substituents, provided the

substituent(s) are not on either carbon adjacent to the carbon C=0 is attached, and each substituent is independently selected from: Ci-C3alkyl, Ci-C3haloalkyl, Ci-C3thiohaloalkyl, Ci-C3alkoxy, C1-Cshaloalkoxy, halogen, NO2, SFs, CN, CONH2, COOH and C(S)NH2;

R3 is Ci-C3alkyl or Ci-C3haloalkyl;

R4 is pyridine, pyrimidine, pyrazine or pyridazine, wherein the pyridine, pyrimidine, pyrazine or pyridazine is optionally substituted with one to three substituents, independently selected, from C1-C3alkyl, Ci-C3haloalkyl, Ci-C3alkoxy, C3-C4cycloalkyl, halogen or hydroxy;

R5 is hydrogen, halogen, CN, Ci-C3alkyl, Ci-C3haloalkyl, C3-C4cycloalkyl, Ci-C3alkoxy, C1-C3haloalkoxy, Ci-C3alkoxycarbonyl, or di(Ci-C3alkoxy)methane; with the proviso that R4 is not pyridin-3-yl, if Ai , A2, A3 and A4 are all CH; ; or a stereoisomer, enantiomer, tautomer and N-oxide of the compound of formula I, or agrochemically acceptable salt thereof.

2. The compound according to claim 1 wherein R3 is methyl.

3. The compound according to either claim 1 or claim 2 wherein Ri is hydrogen; Ci-C6alkyl optionally substituted with one substituent selected from: CN, CONH2, COOH, NO2, and -Si(CH3)3; C1- Cehaloalkyl; C2-C6alkenyl; C2-C6alkynyl; C2-C6haloalkynyl; C3-C4cycloalkyl- Ci-C2alkyl - wherein the C3-C4cycloalkyl- is optionally substituted with 1 or 2 halo atoms; oxetan-3-yl-CH2-; or benzyl optionally substituted with halo or Ci-C3haloalkyl.

The compound according to any one of claims 1 to 3, wherein F¾ is one of Zi to Z10


5. The compound according to any one of claims 1 to 4, wherein Q is selected from Q-1 to Q-12


Q-9 Q-10 Q-11 Q-12

wherein R4 is pyridine, pyrimidine, pyrazine or pyridazine, wherein the pyridine, pyrimidine, pyrazine or pyridazine is optionally substituted with one to three substituents, independently selected, from Ci-C3alkyl, Ci-C3haloalkyl, Ci-C3alkoxy, C3-C4cycloalkyl, halogen or hydroxy.

6. The compound according to any one of claims 1 to 5, wherein R4 is 2-pyridine or 2-pyrimidine optionally substituted by a substituent from halogen and Ci-C3alkoxy.

7. The compound according to claim 6, wherein Ri is cyclopropyl-Chb-, CHºCCH2-, hydrogen, or Me.

8. A composition comprising a compound as defined in any one of claims 1 to 7, one or more auxiliaries and diluent, and optionally one more other active ingredient.

9. A method of combating and controlling insects, acarines, nematodes or molluscs which comprises applying to a pest, to a locus of a pest, or to a plant susceptible to attack by a pest an insecticidally, acaricidally, nematicidally or molluscicidally effective amount of a compound as defined as defined in any one of claims 1 to 7 or a composition as defined claim 8.

10. A method for the protection of plant propagation material from the attack by insects, acarines, nematodes or molluscs, which comprises treating the propagation material or the site, where the propagation material is planted, with an effective amount of a compound as defined in any one of claims 1 to 7 or a composition as defined claim 8.

1 1. A plant propagation material, such as a seed, comprising, or treated with or adhered thereto, a compound as defined in any one of claims 1 to 7 or a composition as defined claim 8.

12. A method of controlling parasites in or on an animal in need thereof comprising administering an effective amount of a compound as defined in any one of claims 1 to 7 or a composition as defined claim 8.