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1. WO2020069353 - COMPOUNDS AND COMPOSITIONS FOR OCULAR DELIVERY

Publication Number WO/2020/069353
Publication Date 02.04.2020
International Application No. PCT/US2019/053513
International Filing Date 27.09.2019
IPC
A61K 31/165 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
16Amides, e.g. hydroxamic acids
165having aromatic rings, e.g. colchicine, atenolol, progabide
C07D 209/04 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
209Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
02condensed with one carbocyclic ring
04Indoles; Hydrogenated indoles
C07D 209/08 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
209Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
02condensed with one carbocyclic ring
04Indoles; Hydrogenated indoles
08with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
CPC
A61K 31/165
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
16Amides, e.g. hydroxamic acids
165having aromatic rings, e.g. colchicine, atenolol, progabide
C07D 209/04
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
209Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
02condensed with one carbocyclic ring
04Indoles; Hydrogenated indoles
C07D 209/08
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
209Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
02condensed with one carbocyclic ring
04Indoles; Hydrogenated indoles
08with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
Applicants
  • GRAYBUG VISION, INC. [US]/[US]
Inventors
  • BAUMAN, John, G.
  • YANG, Ming
  • HOANG, Nu
  • CUNNINGGHAM, Emmett
  • CLELAND, Jeffrey, L.
Agents
  • BELLOWS, Brent, R.
  • KNOWLES, Sherry, M.
  • PROSSER, Anthony, R.
  • STRONG, Katie, L.
Priority Data
62/737,67827.09.2018US
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) COMPOUNDS AND COMPOSITIONS FOR OCULAR DELIVERY
(FR) COMPOSÉS ET COMPOSITIONS POUR ADMINISTRATION OCULAIRE
Abstract
(EN)
The present invention provides new prodrags of Sunitinib, Brinzolamide, and Dorzolamide and compositions to treat medical disorders, for example glaucoma, a disorder or abnormality related to an increase in intraocular pressure (TOP), a disorder requiring neuroprotection, age-related macular degeneration, or diabetic retinopathy.
(FR)
La présente invention concerne de nouveaux promédicaments de Sunitinib, Brinzolamide et Dorzolamide et des compositions pour traiter des troubles médicaux, par exemple le glaucome, un trouble ou une anomalie liés à une augmentation de la pression intraoculaire (TOP), un trouble nécessitant une neuroprotection, la dégénérescence maculaire liée à l'âge ou la rétinopathie diabétique.
Latest bibliographic data on file with the International Bureau