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1. WO2020006329 - SALTS OF (S)-(5-CYCLOBUTOXY-2-METHYL-6-(1-(PIPERIDIN-4-YL)-1H-PYRAZOL-4-YL)-3,4-DIHYDROQUINOLIN-1(2H)-YL)(CYCLOPROPYL)METHANONE AND SOLID FORMS THEREOF

Publication Number WO/2020/006329
Publication Date 02.01.2020
International Application No. PCT/US2019/039677
International Filing Date 28.06.2019
IPC
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
435
having six-membered rings with one nitrogen as the only ring hetero atom
47
Quinolines; Isoquinolines
4709
Non-condensed quinolines containing further heterocyclic rings
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
401
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
14
containing three or more hetero rings
A61K 31/4709 (2006.01)
C07D 401/14 (2006.01)
CPC
A61K 31/4709
C07D 401/14
Applicants
  • FORMA THERAPEUTICS, INC. [US/US]; 500 Arsenal Street Suite 100 Watertown, Massachusetts 02472, US
Inventors
  • LUKE, George P.; US
Agents
  • D'AMATO, Erica M.; US
  • ADATO, Ronen; US
  • AUGST, Alexander; US
  • BUTEAU, Kristen C.; US
  • BYCHOWSKI, Meaghan E.; US
  • DAUKSS, Dana M.; US
  • FORCIER, John V.; US
  • HALEY, Christopher K.; US
  • HAULBROOK, William R.; US
  • HAWVER, Lisa A.; US
  • JARRELL, Brenda Herschbach; US
  • JUDA, Cristin E.; US
  • LI, Bin; US
  • LI, Xiaodong; US
  • LYON, Charles E.; US
  • MA, Longle; US
  • MEDINA, Rolando; US
  • MONG, Surin K.; US
  • MONROE, Margo R.; US
  • PACE, Nicholas J.; US
  • PYSHER, Paul A.; US
  • REARICK, John P.; US
  • REESE, Brian E.; US
  • SAHR, Robert N.; US
  • SCHMITT, Michael; US
  • SCHONEWALD, Stephanie L.; US
  • SHINALL, Michael A.; US
  • SHORE, David E.; US
  • SMITH, Maria C.; US
  • SUH, Su Kyung; US
  • TSE, Janet M.; US
  • VETTER, Michael L.; US
  • VRABLIK, Tracy L.; US
Priority Data
62/692,54629.06.2018US
62/692,55429.06.2018US
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) SALTS OF (S)-(5-CYCLOBUTOXY-2-METHYL-6-(1-(PIPERIDIN-4-YL)-1H-PYRAZOL-4-YL)-3,4-DIHYDROQUINOLIN-1(2H)-YL)(CYCLOPROPYL)METHANONE AND SOLID FORMS THEREOF
(FR) SELS DE (S)-(5-CYCLOBUTOXY-2-MÉTHYL-6-(1- (PIPÉRIDIN-4-YL)-1H-PYRAZOL-4-YL)-3,4-DIHYDROQUINOLIN-1(2H)-YL)(CYCLOPROPYL)MÉTHANONE ET LEURS FORMES SOLIDES
Abstract
(EN)
The present disclosure reports salts of (S)-(5-cyclobutoxy-2-methyl-6-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)-3,4-dihydroquinolin-1(2H)-yl)(cyclopropyl)methanone, solid forms thereof, and methods of making and using the same.
(FR)
La présente invention concerne des sels de (S)-(5-cyclobutoxy-2-méthyl-6-(1-(pipéridin-4-yl)-1H-pyrazol-4-yl)-3,4-dihydroquinolin-1(2H)-yl)(cyclopropyl) méthanone, leurs formes solides, et des procédés de production et d'utilisation de ceux-ci.
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