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1. (WO2019046465) THERAPEUTIC INDOLES
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Pub. No.: WO/2019/046465 International Application No.: PCT/US2018/048607
Publication Date: 07.03.2019 International Filing Date: 29.08.2018
IPC:
A61K 31/166 (2006.01) ,A61K 31/404 (2006.01)
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
16
Amides, e.g. hydroxamic acids
165
having aromatic rings, e.g. colchicine, atenolol, progabide
166
having the carbon atom of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
40
having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
403
condensed with carbocyclic rings, e.g. carbazole
404
Indoles, e.g. pindolol
Applicants:
FREUNDLICH, Joel S. [US/US]; US
ALLAND, David [US/US]; US
NEIDITCH, Matthew B. [US/US]; US
INOYAMA, Daigo [US/US]; US
CAPODAGLI, Glenn [US/US]; US
KUMAR, Pradeep [US/US]; US
RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY [US/US]; Old Queens, Somerset and George Streets New Brunswick, New Jersey 08901, US
Inventors:
FREUNDLICH, Joel S.; US
ALLAND, David; US
NEIDITCH, Matthew B.; US
INOYAMA, Daigo; US
CAPODAGLI, Glenn; US
KUMAR, Pradeep; US
Agent:
HARRIS, Robert J.; US
VIKSNINS, Ann S.; US
MALEN, Peter L.; US
MICKELSON, John W.; US
KRUEGER, Katherine A.D.; US
KLIMA SILBERG, Catherine I.; US
PADYS, Danny J.; US
ANDRUS, Alex; US
Priority Data:
62/551,48229.08.2017US
Title (EN) THERAPEUTIC INDOLES
(FR) INDOLES THÉRAPEUTIQUES
Abstract:
(EN) The invention provides compounds of formula I and salts thereof wherein R1-R4 have any of the meanings described in the specification. The compounds are useful for treating bacterial infections (e.g. tuberculosis).
(FR) La présente invention concerne des composés de formule (I) et leurs sels, R1-R4 ayant l'une quelconque des valeurs définies dans la description. Ces composés sont utiles dans le traitement d'infections bactériennes (par ex., la tuberculose).
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JO, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)