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1. (WO2018226155) COMPOUNDS USEFUL IN INHIBITING HUMAN TREFOIL FACTOR 3
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Pub. No.: WO/2018/226155 International Application No.: PCT/SG2018/050277
Publication Date: 13.12.2018 International Filing Date: 05.06.2018
IPC:
C07D 493/04 (2006.01) ,C07D 491/22 (2006.01) ,A61K 31/519 (2006.01) ,A61K 31/37 (2006.01) ,A61P 35/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
493
Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
02
in which the condensed system contains two hetero rings
04
Ortho-condensed systems
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
491
Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/-C07D459/290
22
in which the condensed system contains four or more hetero rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
495
having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
505
Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
519
ortho- or peri-condensed with heterocyclic rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
335
having oxygen as the only ring hetero atom, e.g. fungichromin
365
Lactones
366
having six-membered rings, e.g. delta-lactones
37
Coumarins, e.g. psoralen
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
35
Antineoplastic agents
Applicants:
NATIONAL UNIVERSITY OF SINGAPORE [SG/SG]; 21 Lower Kent Ridge Road, Singapore 119077, SG
UNIVERSITY OF MYSORE [IN/IN]; Crawford Hall, Mysore, Karnataka 570 005, IN
BANGALORE UNIVERSITY [IN/IN]; Jnana Bharathi Campus, Bengaluru, Karnataka 560056, IN
Inventors:
LOBIE, Peter Edward; SG
PANDEY, Vijay Kumar; SG
KANCHUGARAKOPPAL SUBBEGOWDA, Rangappa; IN
BASAPPA, Basappa; IN
CHAKRABHAVI DHANANJAYA, Mohan; IN
RANGAPPA, Shobith; IN
Agent:
KINNAIRD, James Welsh; SG
Priority Data:
10201704579V05.06.2017SG
Title (EN) COMPOUNDS USEFUL IN INHIBITING HUMAN TREFOIL FACTOR 3
(FR) COMPOSÉS UTILES POUR INHIBER LE FACTEUR 3 EN FEUILLE DE TRÈFLE HUMAIN
Abstract:
(EN) The present invention relates to compounds of Formula I, wherein A, R1 to R6, and x to z are defined herein, and their use in inhibiting Human trefoil factor 3.
(FR) La présente invention concerne des composés de formule I, dans laquelle A, R\ à Rg, et x à z sont tels que définis dans la description, et leur utilisation dans l'inhibition du facteur 3 en feuille de trèfle humain.
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JO, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)