Some content of this application is unavailable at the moment.
If this situation persist, please contact us atFeedback&Contact
1. (WO2018199277) CRYSTAL FORM AND SALT OF 3-(3,5-DICHLORO-4-HYDROXYBENZOYL)-1,1-DIOXO-2,3-DIHYDRO-1,3-BENZOTHIAZOLE
Latest bibliographic data on file with the International Bureau    Submit observation

Pub. No.: WO/2018/199277 International Application No.: PCT/JP2018/017128
Publication Date: 01.11.2018 International Filing Date: 27.04.2018
IPC:
C07D 277/62 (2006.01) ,A61K 31/428 (2006.01) ,A61P 19/06 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
277
Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
60
condensed with carbocyclic rings or ring systems
62
Benzothiazoles
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
41
having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole
425
Thiazoles
428
condensed with carbocyclic rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
19
Drugs for skeletal disorders
06
Antigout agents, e.g. antihyperuricemic or uricosuric agents
Applicants:
株式会社富士薬品 FUJI YAKUHIN CO., LTD. [JP/JP]; 埼玉県さいたま市大宮区桜木町4丁目383番地 4-383, Sakuragi-cho, Omiya-ku, Saitama-shi, Saitama 3309508, JP
Inventors:
雨田 淳一郎 UDA, Junichiro; JP
小橋 精一 KOBASHI, Seiichi; JP
長谷川 美佐 HASEGAWA, Misa; JP
Agent:
高橋 剛 TAKAHASHI, Takeshi; JP
高橋 雅和 TAKAHASHI, Masakazu; JP
高橋 友和 TAKAHASHI, TOMOKAZU; 東京都中央区日本橋3丁目6番10号 マスキチビル3階 3F, Masukichi-Bldg, 6-10, Nihonbashi 3-Chome, Chuo-ku, Tokyo 1030027, JP
Priority Data:
2017-09933428.04.2017JP
Title (EN) CRYSTAL FORM AND SALT OF 3-(3,5-DICHLORO-4-HYDROXYBENZOYL)-1,1-DIOXO-2,3-DIHYDRO-1,3-BENZOTHIAZOLE
(FR) FORME CRISTALLINE ET SEL DE 3-(3,5-DICHLORO-4-HYDROXYBENZOYL)-1,1-DIOXO-2,3-DIHYDRO-1,3-BENZOTHIAZOLE
(JA) 3-(3,5-ジクロロ-4-ヒドロキシベンゾイル)-1,1-ジオキソ-2,3-ジヒドロ-1,3-ベンゾチアゾールの結晶形及び塩
Abstract:
(EN) Provided are: a pharmaceutical composition containing a type I crystal of 3-(3,5-dichloro-4-hydroxybenzoyl)-1,1-dioxo-2,3-dihydro-1,3-benzothiazole, a type II crystal of 3-(3,5-dichloro-4-hydroxybenzoyl)-1,1-dioxo-2,3-dihydro-1,3-benzothiazole, a hydrate of 3-(3,5-dichloro-4-hydroxybenzoyl)-1,1-dioxo-2,3-dihydro-1,3-benzothiazole, a salt thereof, and a pharmaceutically acceptable carrier; and a method for producing the same.
(FR) L'invention concerne : une composition pharmaceutique contenant un cristal de type I de 3-(3,5-dichloro-4-hydroxybenzoyl)-1,1-dioxo-2,3-dihydro-1,3-benzothiazole, un cristal de type II de 3-(3,5-dichloro-4-hydroxybenzoyl)-1,1-dioxo-2,3-dihydro-1,3-benzothiazole, un hydrate de 3-(3,5-dichloro-4-hydroxybenzoyl)-1,1-dioxo-2,3-dihydro-1,3-benzothiazole, un sel de celui-ci, et un véhicule pharmaceutiquement acceptable ; ainsi qu'un procédé de production de celui-ci.
(JA) 3-(3,5-ジクロロ-4-ヒドロキシベンゾイル)-1,1-ジオキソ-2,3-ジヒドロ-1,3-ベンゾチアゾールのI形結晶、3-(3,5-ジクロロ-4-ヒドロキシベンゾイル)-1,1-ジオキソ-2,3-ジヒドロ-1,3-ベンゾチアゾールのII形結晶、3-(3,5-ジクロロ-4-ヒドロキシベンゾイル)-1,1-ジオキソ-2,3-ジヒドロ-1,3-ベンゾチアゾールの水和物、これらの塩、及び薬学的に許容される担体を含有する医薬組成物、ならびにその製造方法。
front page image
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JO, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: Japanese (JA)
Filing Language: Japanese (JA)