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1. WO2018199277 - CRYSTAL FORM AND SALT OF 3-(3,5-DICHLORO-4-HYDROXYBENZOYL)-1,1-DIOXO-2,3-DIHYDRO-1,3-BENZOTHIAZOLE

Publication Number WO/2018/199277
Publication Date 01.11.2018
International Application No. PCT/JP2018/017128
International Filing Date 27.04.2018
IPC
C07D 277/62 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
277Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
60condensed with carbocyclic rings or ring systems
62Benzothiazoles
A61K 31/428 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
41having five-membered rings with two or more ring hetero atoms, at least one of which is nitrogen, e.g. tetrazole
425Thiazoles
428condensed with carbocyclic rings
A61P 19/06 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
19Drugs for skeletal disorders
06Antigout agents, e.g. antihyperuricemic or uricosuric agents
CPC
A61K 31/428
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
41having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
425Thiazoles
428condensed with carbocyclic rings
A61P 19/06
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
19Drugs for skeletal disorders
06Antigout agents, e.g. antihyperuricemic or uricosuric agents
C07B 2200/13
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
2200Indexing scheme relating to specific properties of organic compounds
13Crystalline forms, e.g. polymorphs
C07D 277/62
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
277Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
60condensed with carbocyclic rings or ring-systems
62Benzothiazoles
Applicants
  • 株式会社富士薬品 FUJI YAKUHIN CO., LTD. [JP]/[JP]
Inventors
  • 雨田 淳一郎 UDA, Junichiro
  • 小橋 精一 KOBASHI, Seiichi
  • 長谷川 美佐 HASEGAWA, Misa
Agents
  • 高橋 剛 TAKAHASHI, Takeshi
  • 高橋 雅和 TAKAHASHI, Masakazu
  • 高橋 友和 TAKAHASHI, TOMOKAZU
Priority Data
2017-09933428.04.2017JP
Publication Language Japanese (JA)
Filing Language Japanese (JA)
Designated States
Title
(EN) CRYSTAL FORM AND SALT OF 3-(3,5-DICHLORO-4-HYDROXYBENZOYL)-1,1-DIOXO-2,3-DIHYDRO-1,3-BENZOTHIAZOLE
(FR) FORME CRISTALLINE ET SEL DE 3-(3,5-DICHLORO-4-HYDROXYBENZOYL)-1,1-DIOXO-2,3-DIHYDRO-1,3-BENZOTHIAZOLE
(JA) 3-(3,5-ジクロロ-4-ヒドロキシベンゾイル)-1,1-ジオキソ-2,3-ジヒドロ-1,3-ベンゾチアゾールの結晶形及び塩
Abstract
(EN)
Provided are: a pharmaceutical composition containing a type I crystal of 3-(3,5-dichloro-4-hydroxybenzoyl)-1,1-dioxo-2,3-dihydro-1,3-benzothiazole, a type II crystal of 3-(3,5-dichloro-4-hydroxybenzoyl)-1,1-dioxo-2,3-dihydro-1,3-benzothiazole, a hydrate of 3-(3,5-dichloro-4-hydroxybenzoyl)-1,1-dioxo-2,3-dihydro-1,3-benzothiazole, a salt thereof, and a pharmaceutically acceptable carrier; and a method for producing the same.
(FR)
L'invention concerne : une composition pharmaceutique contenant un cristal de type I de 3-(3,5-dichloro-4-hydroxybenzoyl)-1,1-dioxo-2,3-dihydro-1,3-benzothiazole, un cristal de type II de 3-(3,5-dichloro-4-hydroxybenzoyl)-1,1-dioxo-2,3-dihydro-1,3-benzothiazole, un hydrate de 3-(3,5-dichloro-4-hydroxybenzoyl)-1,1-dioxo-2,3-dihydro-1,3-benzothiazole, un sel de celui-ci, et un véhicule pharmaceutiquement acceptable ; ainsi qu'un procédé de production de celui-ci.
(JA)
3-(3,5-ジクロロ-4-ヒドロキシベンゾイル)-1,1-ジオキソ-2,3-ジヒドロ-1,3-ベンゾチアゾールのI形結晶、3-(3,5-ジクロロ-4-ヒドロキシベンゾイル)-1,1-ジオキソ-2,3-ジヒドロ-1,3-ベンゾチアゾールのII形結晶、3-(3,5-ジクロロ-4-ヒドロキシベンゾイル)-1,1-ジオキソ-2,3-ジヒドロ-1,3-ベンゾチアゾールの水和物、これらの塩、及び薬学的に許容される担体を含有する医薬組成物、ならびにその製造方法。
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