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1. (WO2018160024) PIPERIDINE-ARYL DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT
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Pub. No.: WO/2018/160024 International Application No.: PCT/KR2018/002508
Publication Date: 07.09.2018 International Filing Date: 28.02.2018
IPC:
C07D 401/12 (2006.01) ,A61K 31/444 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
401
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02
containing two hetero rings
12
linked by a chain containing hetero atoms as chain links
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
435
having six-membered rings with one nitrogen as the only ring hetero atom
44
Non-condensed pyridines; Hydrogenated derivatives thereof
4427
containing further heterocyclic ring systems
444
containing a six-membered ring with nitrogen as a ring hetero atom, e.g. amrinone
Applicants:
한국화학연구원 KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY [KR/KR]; 대전시 유성구 가정로 141 141, Gajeong-ro, Yuseong-gu, Daejeon 34114, KR
경북대학교 산학협력단 KYUNGPOOK NATIONAL UNIVERSITY INDUSTRY-ACADEMIC COOPERATION FOUNDATION [KR/KR]; 대구시 북구 대학로 80 80, Daehak-ro, Buk-gu, Daegu 41566, KR
경북대학교병원 KYUNGPOOK NATIONAL UNIVERSITY HOSPITAL [KR/KR]; 대구시 중구 동덕로 130 130, Dongdeok-ro, Jung-gu, Daegu 41944, KR
광주과학기술원 GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY [KR/KR]; 광주시 북구 첨단과기로 123 123, Cheomdangwagi-ro, Buk-gu, Gwangju 61005, KR
Inventors:
안진희 AHN, Jin Hee; KR
배은정 BAE, Eun Jung; KR
이인규 LEE, In-Kyu; KR
전재한 JEON, Jae-Han; KR
강승규 KANG, Seung Kyu; KR
이규명 LEE, Kyu-Myung; KR
정관령 JEONG, Kwan Young; KR
장윤경 JANG, Yoon Kyung; KR
김광록 KIM, Kwang-Rok; KR
이상달 RHEE, Sang Dal; KR
배명애 BAE, Myung-Ae; KR
김효진 KIM, Hyojin; KR
Agent:
손민 SON, Min; KR
Priority Data:
10-2017-002681228.02.2017KR
Title (EN) PIPERIDINE-ARYL DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT
(FR) DÉRIVÉ DE PIPÉRIDINE-ARYLE OU SEL PHARMACEUTIQUEMENT ACCEPTABLE DE CELUI-CI, SON PROCÉDÉ DE PRÉPARATION ET COMPOSITION PHARMACEUTIQUE CONTENANT CELUI-CI EN TANT QUE PRINCIPE ACTIF
(KO) 피페리딘-아릴 유도체 또는 이의 약학적으로 허용 가능한 염, 이의 제조방법, 및 이를 유효성분으로 함유하는 약제학적 조성물
Abstract:
(EN) The present invention relates to: a piperidine-aryl derivative having G-protein-coupled receptor (G-protein-coupled receptor 119; GPR119) agonist activity, or a pharmaceutically acceptable salt thereof; a method for preparing same; and a pharmaceutical composition containing same as an active ingredient.
(FR) La présente invention concerne : un dérivé de pipéridine-aryle ayant une activité agoniste vis-à-vis du récepteur couplé à la protéine G (G-protein-coupled receptor 119 ; GPR119), ou un sel pharmaceutiquement acceptable de celui-ci ; son procédé de préparation ; et une composition pharmaceutique le contenant en tant que principe actif.
(KO) 본 발명은 G 단백질 결합 수용체(Gprotein-coupled receptor 119; GPR119) 항진 활성을 가지는 피페리딘-아릴 유도체 또는 이의 약제학적으로 허용 가능한 염; 이의 제조방법; 및 이를 유효성분으로 함유하는 약제학적 조성물에 관한 것이다.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JO, JP, KE, KG, KH, KN, KP, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: Korean (KO)
Filing Language: Korean (KO)