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1. (WO2018080072) NOVEL MACROLIDE-BASED COMPOUND, METHOD FOR PRODUCING SAME, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING MALARIA AND CONTAINING SAME AS ACTIVE INGREDIENT
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Pub. No.: WO/2018/080072 International Application No.: PCT/KR2017/011396
Publication Date: 03.05.2018 International Filing Date: 16.10.2017
IPC:
C07H 17/08 (2006.01) ,A61K 31/70 (2006.01) ,C12N 1/20 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
H
SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
17
Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
04
Heterocyclic radicals containing only oxygen as ring hetero atoms
08
Hetero rings containing eight or more ring members, e.g. erythromycins
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
70
Carbohydrates; Sugars; Derivatives thereof
C CHEMISTRY; METALLURGY
12
BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
N
MICRO-ORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICRO-ORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
1
Micro-organisms, e.g. protozoa; Compositions thereof; Processes of propagating, maintaining or preserving micro-organisms or compositions thereof; Processes of preparing or isolating a composition containing a micro-organism; Culture media therefor
20
Bacteria; Culture media therefor
Applicants:
한국생명공학연구원 KOREA RESEARCH INSTITUTE OF BIOSCIENCE AND BIOTECHNOLOGY [KR/KR]; 대전시 유성구 과학로 125 125, Gwahak-ro Yuseong-gu Daejeon 34141, KR
Inventors:
안종석 AHN, Jong Seog; KR
장재혁 JANG, Jae-Hyuk; KR
고성균 KO, Sung-Kyun; KR
류인자 RYOO, In Ja; KR
손상근 SON, Sang Keun; KR
김보연 KIM, Bo Yeon; KR
성낙균 SOUNG, Nak Kyun; KR
이경호 LEE, Kyung Ho; KR
홍영수 HONG, Young-Soo; KR
Agent:
특허법인주원 B & IP-JOOWON PATENT AND LAW FIRM; KR
Priority Data:
10-2016-014089827.10.2016KR
10-2017-012850902.10.2017KR
Title (EN) NOVEL MACROLIDE-BASED COMPOUND, METHOD FOR PRODUCING SAME, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING MALARIA AND CONTAINING SAME AS ACTIVE INGREDIENT
(FR) NOUVEAU COMPOSÉ À BASE DE MACROLIDE, SON PROCÉDÉ DE PRODUCTION, ET COMPOSITION PHARMACEUTIQUE DESTINÉE À PRÉVENIR OU À TRAITER LE PALUDISME ET LE CONTENANT À TITRE DE PRINCIPE ACTIF
(KO) 신규한 매크로라이드계 화합물, 이의 제조방법 및 이를 유효성분으로 함유하는 말라리아의 예방 또는 치료용 약학적 조성물
Abstract:
(EN) The present invention relates to a novel macrolide-based compound, a method for producing the same, and a pharmaceutical composition, which is for preventing or treating malaria and contains the novel macrolide-based compound as an active ingredient. The macrolide-based compound represented by chemical formula 1 according to the present invention effectively exhibits an antiprotozoal activity against Plasmodium sp. protozoan, and thus can be usefully used to prevent or treat malaria.
(FR) La présente invention concerne un nouveau composé à base de macrolide, son procédé de production, et une composition pharmaceutique, qui est destinée à prévenir ou à traiter le paludisme et le contenant à titre de principe actif. Le composé à base de macrolide représenté par la formule chimique 1 selon la présente invention présente une activité antiprotozoaire efficace contre le protozoaire Plasmodium sp., et peut par conséquent être utilisé de manière utile pour prévenir ou traiter le paludisme.
(KO) 본 발명은 신규한 매크로라이드계 화합물, 이의 제조방법 및 이를 유효성분으로 함유하는 말라리아의 예방 또는 치료용 약학적 조성물에 관한 것으로, 본 발명에 따른 화학식 1로 표시되는 매크로라이드계 화합물은 플라스모듐 속(Plasmodium sp.) 원충에 대하여 항원충 활성을 효과적으로 나타내어 말라리아의 예방 또는 치료에 유용하게 사용될 수 있는 효과가 있다.
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JO, JP, KE, KG, KH, KN, KP, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: Korean (KO)
Filing Language: Korean (KO)