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1. (WO2018052035) DIARYL AZOLE COMPOUND AND PESTICIDE
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Pub. No.: WO/2018/052035 International Application No.: PCT/JP2017/033103
Publication Date: 22.03.2018 International Filing Date: 13.09.2017
IPC:
C07D 233/64 (2006.01) ,A01N 25/04 (2006.01) ,A01N 43/50 (2006.01) ,A01N 43/54 (2006.01) ,A01N 43/56 (2006.01) ,A01N 43/653 (2006.01) ,A01N 43/78 (2006.01) ,A01N 43/824 (2006.01) ,A01P 7/02 (2006.01) ,A01P 7/04 (2006.01) ,A61K 31/4439 (2006.01) ,A61K 31/506 (2006.01) ,A61P 31/10 (2006.01) ,A61P 31/14 (2006.01) ,C07D 401/04 (2006.01) ,C07D 401/14 (2006.01) ,C07D 403/04 (2006.01) ,C07D 403/10 (2006.01) ,C07D 403/14 (2006.01) ,C07D 413/10 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
233
Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
54
having two double bonds between ring members or between ring members and non-ring members
64
with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
N
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
25
Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
02
containing liquids as carriers, diluents or solvents
04
Dispersions or gels
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
N
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43
Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
48
having rings with two nitrogen atoms as the only ring hetero atoms
50
1,3-Diazoles; Hydrogenated 1,3-diazoles
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
N
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43
Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
48
having rings with two nitrogen atoms as the only ring hetero atoms
54
1,3-Diazines; Hydrogenated 1,3-diazines
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
N
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43
Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
48
having rings with two nitrogen atoms as the only ring hetero atoms
56
1,2-Diazoles; Hydrogenated 1,2-diazoles
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
N
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43
Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
64
having rings with three nitrogen atoms as the only ring hetero atoms
647
Triazoles; Hydrogenated triazoles
653
1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
N
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43
Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
72
having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms
74
five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
78
1,3-Thiazoles; Hydrogenated 1,3-thiazoles
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
N
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43
Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
72
having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms
82
five-membered rings with three hetero atoms
824
1,3,4-Oxa(thia)diazoles; Hydrogenated 1,3,4-oxa(thia)diazoles
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
P
BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
7
Arthropodicides
02
Acaricides
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
P
BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
7
Arthropodicides
04
Insecticides
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
435
having six-membered rings with one nitrogen as the only ring hetero atom
44
Non-condensed pyridines; Hydrogenated derivatives thereof
4427
containing further heterocyclic ring systems
4439
containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
495
having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
505
Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
506
not condensed and containing further heterocyclic rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
31
Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
10
Antimycotics
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
31
Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
12
Antivirals
14
for RNA viruses
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
401
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02
containing two hetero rings
04
directly linked by a ring-member-to-ring- member bond
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
401
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
14
containing three or more hetero rings
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
403
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/167
02
containing two hetero rings
04
directly linked by a ring-member-to-ring- member bond
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
403
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/167
02
containing two hetero rings
10
linked by a carbon chain containing aromatic rings
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
403
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/167
14
containing three or more hetero rings
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
413
Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
02
containing two hetero rings
10
linked by a carbon chain containing aromatic rings
Applicants:
日本曹達株式会社 NIPPON SODA CO., LTD. [JP/JP]; 東京都千代田区大手町二丁目2番1号 2-1, Ohtemachi 2-chome, Chiyoda-ku, Tokyo 1008165, JP
Inventors:
阪西 慶太 SAKANISHI Keita; JP
岩佐 孝男 IWASA Takao; JP
青山 光 AOYAMA Hikaru; JP
崎山 訓史 SAKIYAMA Norifumi; JP
牛島 大佑 USHIJIMA Daisuke; JP
松井 麻記 MATSUI Maki; JP
小林 朝巳 KOBAYASHI Tomomi; JP
Agent:
志賀 正武 SHIGA Masatake; JP
高橋 詔男 TAKAHASHI Norio; JP
鈴木 三義 SUZUKI Mitsuyoshi; JP
村山 靖彦 MURAYAMA Yasuhiko; JP
Priority Data:
2016-18046715.09.2016JP
2017-08926628.04.2017JP
Title (EN) DIARYL AZOLE COMPOUND AND PESTICIDE
(FR) COMPOSÉ DE DIARYL AZOLE ET PESTICIDE
(JA) ジアリールアゾール化合物および有害生物防除剤
Abstract:
(EN) Provided is a compound represented by formula (I), or a salt thereof. [Formula 1] In formula (I), R1 represents an unsubstituted or substituted C1–6 alkylthio group or the like. A1 represents a nitrogen atom or CH. A2 represents a nitrogen atom or CR2. R2 and R3 each independently represent a hydrogen atom, an unsubstituted or substituted C6–10 aryl group, an unsubstituted or substituted three- to six-member heterocyclic group, or the like. B1 and B2 each independently represent a nitrogen atom or CR5. However, B1 and B2 cannot both be CR5. R5 represents a hydrogen atom, an unsubstituted or substituted C1–6 alkyl group, or the like. R4 represents an unsubstituted or substituted C1–6 alkyl group or the like. R4 is bonded to any one nitrogen atom from among the nitrogen atoms constituting an imidazole ring or a triazole ring. Ar represents an unsubstituted or substituted C6–10 aryl group or the like.
(FR) L'invention concerne un composé représenté par la formule (I), ou un sel de celui-ci. [Formule 1] Dans la formule (I), R 1 représente un groupe alkylthio en C1 – 6 non substitué ou substitué ou similaire. A 1 représente un atome d'azote ou CH. A 2 représente un atome d'azote ou CR 2 . R 2 et R 3 représentent chacun indépendamment un atome d'hydrogène, un groupe aryle en C6-10 non substitué ou substitué, un groupe hétérocyclique à trois jusqu'à six chaînons non substitué ou substitué, ou similaire. B 1 et B 2 représentent chacun indépendamment un atome d'azote ou CR 5 . Cependant, B 1 et B 2 ne peuvent pas être à la fois CR 5 . R 5 représente un atome d'hydrogène, un groupe alkyle en C1-6 non substitué ou substitué, ou similaire. R 4 représente un groupe alkyle en C1-6 non substitué ou substitué ou similaire. R 4 est lié à un atome d'azote quelconque parmi les atomes d'azote constituant un cycle imidazole ou un cycle triazole. Ar représente un groupe aryle en C6-10 non substitué ou substitué ou similaire.
(JA) 式(I)で表される化合物またはその塩。 [化1] 式(I)中、Rは、無置換のもしくは置換基を有するC1~6アルキルチオ基などを示す。Aは、窒素原子またはCHを示す。Aは、窒素原子またはCRを示す。RおよびRは、それぞれ独立に、水素原子、無置換のもしくは置換基を有するC6~10アリール基、または無置換のもしくは置換基を有する3~6員ヘテロシクリル基などを示す。BおよびBは、それぞれ独立に、窒素原子またはCRを示す。但し、BとBがともにCRであることはない。ここで、Rは、水素原子、無置換のもしくは置換基を有するC1~6アルキル基などを示す。Rは、無置換のもしくは置換基を有するC1~6アルキル基などを示す。Rは、イミダゾール環若しくはトリアゾール環を構成する窒素原子のうちのいずれか一つの窒素原子に結合する。Arは、無置換のもしくは置換基を有するC6~10アリール基などを示す。
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JO, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: Japanese (JA)
Filing Language: Japanese (JA)