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1. (WO2018050046) FUSED TRICYCLIC Γ-AMINO ACID DERIVATIVE, PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF
Latest bibliographic data on file with the International Bureau    Submit observation

Pub. No.: WO/2018/050046 International Application No.: PCT/CN2017/101364
Publication Date: 22.03.2018 International Filing Date: 12.09.2017
IPC:
C07C 229/28 (2006.01) ,A61K 31/195 (2006.01) ,A61P 25/04 (2006.01) ,A61P 25/06 (2006.01) ,A61P 29/00 (2006.01)
Applicants: SICHUAN HAISCO PHARMACEUTICAL CO., LTD.[CN/CN]; No.136 Beverley Road, Across The Taiwan Strait Technology Industry Development Park Wenjiang District Chengdu, Sichuan 611130, CN
Inventors: LI, Yao; CN
SHI, Zongjun; CN
XU, Bo; CN
Agent: BEIJING SANYOU INTELLECTUAL PROPERTY AGENCY LTD.; 16th Fl., Block A Corporate Square, No.35 Jinrong Street Beijing 100033, CN
Priority Data:
201610825611.914.09.2016CN
Title (EN) FUSED TRICYCLIC Γ-AMINO ACID DERIVATIVE, PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF
(FR) DÉRIVÉ D'ACIDE Γ-AMINÉ TRICYCLIQUE FUSIONNÉ, SON PROCÉDÉ DE PRÉPARATION ET SON UTILISATION MÉDICALE
(ZH) 稠合三环γ-氨基酸衍生物及其制备方法和在医药上的应用
Abstract: front page image
(EN) Disclosed are a fused tricyclic γ-amino acid derivative and a medical use thereof, in particular, the present invention relates to a fused cyclic γ-amino acid derivative as shown in general formula (I), or a stereoisomer, solvate, metabolite, prodrug, pharmaceutically acceptable salt or eutectic thereof, a pharmaceutical composition containing same, and the use of a compound or the composition in the field of analgesia, wherein the definitions of each substituent in general formula (I) are the same as the definitions in the description.
(FR) L'invention concerne un dérivé d'acide γ-aminé tricyclique fusionné et son utilisation médicale, en particulier, la présente invention concerne un dérivé d'acide gamma-aminé cyclique fusionné tel que représenté dans la formule générale (I), ou un stéréoisomère, un solvate, un métabolite, un promédicament, un sel pharmaceutiquement acceptable ou un eutectique de celui-ci, une composition pharmaceutique le contenant, et l'utilisation d'un composé ou de la composition dans le domaine de l'analgésie, les définitions de chaque substituant dans la formule générale (I) étant les mêmes que les définitions dans la description.
(ZH) 公开了一种稠合三环γ-氨基酸衍生物及其在医药上的应用,具体而言涉及如通式(I)所示的稠合环γ-氨基酸衍生物,或者其立体异构体、溶剂化物、代谢产物、前药、药学上可接受的盐或共晶,包含其的药物组合物以及化合物或组合物在镇痛领域的用途,其中,通式(I)中各取代基的定义与说明书的定义相同。
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JO, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: Chinese (ZH)
Filing Language: Chinese (ZH)