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1. (WO2018011578) METHOD FOR PRODUCING A POLYMORPHIC FORM OF 3-[5-AMINO-4-(3-CYANOBENZOYL)-PYRAZOL-1-YL]-N-CYCLOPROPYL-4-METHYLBENZAMIDE
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Pub. No.: WO/2018/011578 International Application No.: PCT/GB2017/052055
Publication Date: 18.01.2018 International Filing Date: 13.07.2017
IPC:
C07D 231/38 (2006.01) ,A61K 31/415 (2006.01) ,A61P 29/00 (2006.01)
Applicants: MEREO BIOPHARMA 1 LIMITED; 1 Cavendish Place London Greater London W1G 0QF, GB
Inventors: SULEIMAN, Osama; GB
PEREZ, Lucia Romero; GB
HARLACHER, Cornelius Stephan; CH
JONES, Stewart; GB
Agent: GILL JENNINGS & EVERY LLP; The Broadgate Tower 20 Primrose Street London, Greater London EC2A 2ES, GB
CLARKE, Lionel Paul; GB
Priority Data:
1612238.414.07.2016GB
Title (EN) METHOD FOR PRODUCING A POLYMORPHIC FORM OF 3-[5-AMINO-4-(3-CYANOBENZOYL)-PYRAZOL-1-YL]-N-CYCLOPROPYL-4-METHYLBENZAMIDE
(FR) PROCÉDÉ DE PRODUCTION D'UNE FORME POLYMORPHE DE 3- [5-AMINO-4-(3-CYANOBENZOYL)-PYRAZOL-1-YL]-N-CYCLOPROPYL-4-MÉTHYLBENZAMIDE
Abstract:
(EN) This invention relates to a process for the preparation of Form B of 3-[5-amino-4-(3- cyanobenzoyl)-pyrazol-1-yl]-N-cyclopropyl-4-methylbenzamide. Also disclosed herein is Form B of 3-[5-amino-4-(3-cyanobenzoyl)-pyrazol-1-yl]-N-cyclopropyl-4- methylbenzamide, or pharmaceutical compositions thereof, obtainable by the process described herein.
(FR) L'invention concerne un procédé de préparation de la forme B de 3- [5-amino-4-(3-cyanobenzoyl)-pyrazol-1-yl]-N-cyclopropyl-4-méthylbenzamide. L'invention concerne également la forme B de 3- [5-amino-4-(3-cyanobenzoyle)-pyrazol-1-yl]-N-cyclopropyl-4-méthylbenzamide, ou des compositions pharmaceutiques de celui-ci, pouvant être obtenues par le procédé décrit ici.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JO, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)