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1. (WO2018003980) CRYSTAL OF ACID ADDITION SALT OF AMINOCARBOXYLIC ACID, AND METHOD FOR PRODUCING SAME
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Pub. No.: WO/2018/003980 International Application No.: PCT/JP2017/024180
Publication Date: 04.01.2018 International Filing Date: 30.06.2017
IPC:
C07C 211/25 (2006.01) ,A61K 31/195 (2006.01) ,A61P 25/04 (2006.01) ,C07C 309/29 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
211
Compounds containing amino groups bound to a carbon skeleton
01
having amino groups bound to acyclic carbon atoms
25
of an unsaturated carbon skeleton containing rings other than six-membered aromatic rings
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
185
Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
19
Carboxylic acids, e.g. valproic acid
195
having an amino group
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25
Drugs for disorders of the nervous system
04
Centrally acting analgesics, e.g. opioids
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
309
Sulfonic acids; Halides, esters, or anhydrides thereof
01
Sulfonic acids
28
having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
29
of non-condensed six-membered aromatic rings
Applicants:
第一三共株式会社 DAIICHI SANKYO COMPANY,LIMITED [JP/JP]; 東京都中央区日本橋本町三丁目5番1号 3-5-1,Nihonbashi Honcho,Chuo-ku, Tokyo 1038426, JP
Inventors:
沼上 英治 NUMAGAMI, Eiji; JP
東海林 正寛 SHOJI, Masahiro; JP
鈴木 徹也 SUZUKI, Tetsuya; JP
Agent:
石橋 公樹 ISHIBASHI, Koki; JP
竹元 利泰 TAKEMOTO, Toshiyasu; JP
Priority Data:
2016-13132501.07.2016JP
Title (EN) CRYSTAL OF ACID ADDITION SALT OF AMINOCARBOXYLIC ACID, AND METHOD FOR PRODUCING SAME
(FR) CRISTAUX DE SEL D’ADDITION ACIDE D’ACIDE AMINOCARBOXYLIQUE, ET PROCÉDÉ DE FABRICATION DE CEUX-CI
(JA) アミノカルボン酸の酸付加塩の結晶とその製造方法
Abstract:
(EN) The present invention addresses the problem of providing a crystal of a pharmacologically acceptable salt of a bicyclic aminocarboxylic acid derivative. The solution is a crystal of [(1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid-(benzenesulfonate) salt.
(FR) L’invention a pour objet de fournir des cristaux d’un sel pharmacologiquement acceptable d’un dérivé d’acide aminocarboxylique bicyclique. Plus précisément, l’invention concerne des cristaux d’un sel d’acide [(1R,5S,6S)-6-(aminométhyl)-3-éthylbicylco[3.2.0] hept-3-én-6-yl] acétique一(acide benzène sulfonique).
(JA) 本発明の課題は、二環性アミノカルボン酸誘導体の薬理学的に許容される塩の結晶を提供することである。 解決手段は、[(1R,5S,6S)-6-(アミノメチル)-3-エチルビシクロ[3.2.0]ヘプト-3-エン-6-イル]酢酸一(ベンゼンスルホン酸)塩の結晶である。
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JO, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: Japanese (JA)
Filing Language: Japanese (JA)