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1. (WO2017191650) PROCESS FOR THE PREPARATION OF 5-[[[(2S)-2-AMINO-3-[4-(AMINOCARBONYL)-2,6-DIMETHYLPHENYL]-1-OXOPROPYL][(1S)-1-(4-PHENYL-1H-IMIDAZOL-2-YL)ETHYL]AMINO]METHYL-2-METHOXYBENZOIC ACID AND ITS POLYMORPHS THEREOF
Latest bibliographic data on file with the International Bureau    Submit observation

Pub. No.:    WO/2017/191650    International Application No.:    PCT/IN2017/000098
Publication Date: 09.11.2017 International Filing Date: 02.05.2017
IPC:
C07D 233/00 (2006.01), A61K 31/4178 (2006.01), A61P 1/00 (2006.01), C07D 233/64 (2006.01)
Applicants: MSN LABORATORIES PRIVATE LIMITED [IN/IN]; Sy.no.317 & 323 Rudraram (vil), Patancheru (Mdl), Medak (Dist), Hyderabad, Telangana (IN).
THIRUMALAI RAJAN, Srinivasan [IN/IN]; (IN).
ESWARAIAH, Sajja [IN/IN]; (IN).
RAJESHWAR REDDY, Sagyam [IN/IN]; (IN).
PRABHAKAR, Macharla [IN/IN]; (IN).
RAJESHAM, Boge [IN/IN]; (IN)
Inventors: THIRUMALAI RAJAN, Srinivasan; (IN).
ESWARAIAH, Sajja; (IN).
RAJESHWAR REDDY, Sagyam; (IN).
PRABHAKAR, Macharla; (IN).
RAJESHAM, Boge; (IN)
Common
Representative:
THIRUMALAI RAJAN, Srinivasan; (IN)
Priority Data:
201641015345 03.05.2016 IN
201641023195 06.07.2016 IN
201741002480 23.01.2017 IN
201741002481 23.01.2017 IN
Title (EN) PROCESS FOR THE PREPARATION OF 5-[[[(2S)-2-AMINO-3-[4-(AMINOCARBONYL)-2,6-DIMETHYLPHENYL]-1-OXOPROPYL][(1S)-1-(4-PHENYL-1H-IMIDAZOL-2-YL)ETHYL]AMINO]METHYL-2-METHOXYBENZOIC ACID AND ITS POLYMORPHS THEREOF
(FR) PROCÉDÉ DE PRÉPARATION DE L'ACIDE 5-[[[(2S)-2-AMINO-3-[4-(AMINOCARBONYL)-2,6-DIMÉTHYLPHÉNYL]-1-OXOPROPYL][(1S)-1-(4-PHÉNYL-1H-IMIDAZOL-2-YL)ÉTHYL]AMINO]MÉTHYL-2-MÉTHOXYBENZOÏQUE ET SES POLYMORPHES
Abstract: front page image
(EN)The present invention relates to an improved process for the preparation of 5-[[[(2S)-2-amino-3-[4-(aminocarbonyl)-2,6-dimethylphenyl]- l -oxopropyl][(l S)-l -(4-phenyl-l H-imidazol-2-yl)ethyl]amino]methyl]-2-methoxybenzoic acid compound of formula-1, and polymorphs thereof, the compound of formula- 1 is further represented by the following structural formula:
(FR)La présente invention concerne un procédé amélioré de préparation d'acide 5-[[[(2S)-2-amino-3-[4-(aminocarbonyl)-2,6-diméthylphényl]-1-oxopropyl][(1S)-1-(4-phényl-1H-imidazol-2-yl)éthyl]amino]méthyl]-2-méthoxybenzoïque de formule 1, et des polymorphes de celui-ci, le composé de formule 1 étant en outre représenté par la formule structurale suivante :
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)