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1. (WO2017181948) SUBSTITUTED OXAZOLIDONE AND APPLICATION THEREOF
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Pub. No.: WO/2017/181948 International Application No.: PCT/CN2017/081010
Publication Date: 26.10.2017 International Filing Date: 19.04.2017
IPC:
C07F 9/6558 (2006.01) ,A61K 31/675 (2006.01) ,A61P 31/04 (2006.01) ,A61P 31/06 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
F
ACYCLIC, CARBOCYCLIC, OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
9
Compounds containing elements of the 5th Group of the Periodic System
02
Phosphorus compounds
547
Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
6558
containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
66
Phosphorus compounds
675
having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
31
Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
04
Antibacterial agents
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
31
Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
04
Antibacterial agents
06
for tuberculosis
Applicants:
深圳市塔吉瑞生物医药有限公司 SHENZHEN TARGETRX, INC. [CN/CN]; 中国广东省深圳 南山区科苑路15号科兴科学园A1栋301 Room 301, Building A1, Kexing Science Park No. 15 of Keyuan Road, Nanshan District Shenzhen, Guangdong 5180057, CN
Inventors:
王义汉 WANG, Yihan; CN
邢青峰 XING, Qingfeng; CN
Priority Data:
201610255282.922.04.2016CN
Title (EN) SUBSTITUTED OXAZOLIDONE AND APPLICATION THEREOF
(FR) OXAZOLIDONE SUBSTITUÉE ET SON APPLICATION
(ZH) 取代的恶唑烷酮化合物及其应用
Abstract:
(EN) An oxazolidone compound represented by formula (I), or a crystalline form, pharmaceutically acceptable salt, prodrug, metabolite, stereoisomer, isotopic isomer, hydrate, or solvate thereof, and a pharmaceutical composition comprising the compound. The compound has demonstrated inhibitory activity against a broad spectrum of bacteria and low toxicity, and can be used to prepare an antibiotic.
(FR) L'invention concerne un composé d'oxazolidone de formule (I), ou une forme cristalline correspondante, un sel pharmaceutiquement acceptable, un promédicament, un métabolite, un stéréoisomère, un isomère isotopique, un hydrate ou un solvate correspondant, et une composition pharmaceutique comprenant le composé. Le composé a démontré une activité inhibitrice vis-à-vis d'un large spectre de bactéries et une faible toxicité, et il peut être utilisé pour préparer un antibiotique.
(ZH) 式(I)所示的恶唑烷酮化合物,或其晶型、药学上可接受的盐、前药、代谢物、立体异构体、同位素变体、水合物或溶剂合物,包含该化合物的药物组合物。该化合物显示对广谱菌的抑制活性和低毒性,可作为抗生素。
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: Chinese (ZH)
Filing Language: Chinese (ZH)