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1. (WO2017168448) SILICON INCORPORATED QUINOLINES WITH ANTI-MALARIAL AND ANTI-TOXOPLASMOSIS ACTIVITY
Latest bibliographic data on file with the International Bureau    Submit observation

Pub. No.: WO/2017/168448 International Application No.: PCT/IN2017/050118
Publication Date: 05.10.2017 International Filing Date: 30.03.2017
IPC:
A61K 31/47 (2006.01) ,C07D 215/52 (2006.01) ,C07F 7/08 (2006.01)
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
435
having six-membered rings with one nitrogen as the only ring hetero atom
47
Quinolines; Isoquinolines
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
215
Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
02
having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
16
with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
48
Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
50
attached in position 4
52
with aryl radicals attached in position 2
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
F
ACYCLIC, CARBOCYCLIC, OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
7
Compounds containing elements of the 4th Group of the Periodic System
02
Silicon compounds
08
Compounds having one or more C-Si linkages
Applicants: COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH[IN/IN]; Anusandhan Bhawan, Rafi Marg, New Delhi 110001, IN
Inventors: REDDY, Dumbala Srinivasa; IN
SHANMUGAM, Dhanasekaran; IN
RAMESH, Remya; IN
SHUKLA, Anurag; IN
BELEKAR, Meenakshi Anil; IN
Agent: KOUL, Sunaina; IN
SALHOTRA, Anuradha; IN
DHAWAN, Ramesh Chander; IN
GARG, Avi; IN
PRASAD, Suman Lata; IN
MAHAJAN, Bharti; IN
SHARMA, Nidhi; IN
Priority Data:
20161101107030.03.2016IN
Title (EN) SILICON INCORPORATED QUINOLINES WITH ANTI-MALARIAL AND ANTI-TOXOPLASMOSIS ACTIVITY
(FR) QUINOLÉINES À SILICIUM INCORPORÉ PRÉSENTANT UNE ACTIVITÉ ANTI-PALUDÉENNE ET ANTI-TOXOPLASMOSE
Abstract:
(EN) The present invention discloses a silicon incorporated quinoline of formula (I) wherein, X, Y, A, R1 and R2 are as described. The present invention further discloses a process for the preparation of silicon incorporated quinolines of formula I; a pharmaceutical composition comprising silicon incorporated quinolines of formula (I) or pharmaceutically acceptable salt thereof. The present invention also discloses a method for treating diseases caused by Plasmodium falciparum or other coccidian parasites using the silicon incorporated quinolines of formula I or pharmaceutically acceptable salt thereof.
(FR) La présente invention concerne une quinoléine à silicium incorporé de formule (I) dans laquelle X, Y, A, R1 et R2 sont tels que décrits. La présente invention concerne en outre un procédé pour la préparation de quinoléines à silicium incorporé de formule I ; une composition pharmaceutique comprenant des quinoléines à silicium incorporé de formule (I) ou un sel pharmaceutiquement acceptable de ces dernières. La présente invention concerne également un procédé de traitement de maladies provoquées par Plasmodium falciparum ou d'autres parasites coccidiens à l'aide des quinoléines à silicium incorporé de formule I ou de leurs sels pharmaceutiquement acceptables.
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)