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1. (WO2017156265) DIRECT PALLADIUM-CATALYZED AROMATIC FLUORINATION
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Pub. No.: WO/2017/156265 International Application No.: PCT/US2017/021563
Publication Date: 14.09.2017 International Filing Date: 09.03.2017
IPC:
C07D 471/04 (2006.01) ,B01J 23/44 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
471
Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/-C07D463/251
02
in which the condensed system contains two hetero rings
04
Ortho-condensed systems
B PERFORMING OPERATIONS; TRANSPORTING
01
PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
J
CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS, COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
23
Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/113
38
of noble metals
40
of the platinum group metals
44
Palladium
Applicants:
PRESIDENT AND FELLOWS OF HARVARD COLLEGE [US/US]; 17 Quincy Street Cambridge, MA 02138, US
STUDIENGESELLSCHAFT KOHLE MBH [DE/DE]; Kaiser-Wilhelm-Platz 1 D-45470 Mülheim An Der Ruhr, DE
Inventors:
RITTER, Tobias; DE
GARBER, Jeffrey; DE
YAMAMOTO, Kumiko; JP
Agent:
BAKER, Hunter C.; US
Priority Data:
62/305,71109.03.2016US
62/346,32606.06.2016US
Title (EN) DIRECT PALLADIUM-CATALYZED AROMATIC FLUORINATION
(FR) FLUORATION AROMATIQUE DIRECTE CATALYSÉE PAR DU PALLADIUM
Abstract:
(EN) Provided herein are palladium complexes comprising a ligand of Formula (Α') and a ligand of Formula (B), wherein R1-R18 are as defined herein. The palladium complexes are useful in methods of fluorinating aryl and heteroaryl substrates. Further provided are compositions and kits comprising the palladium complexes.
(FR) L'invention concerne des complexes de palladium comprenant un ligand de formule (Α') et un ligand de formule (B) dans lesquelles R1 à R18 sont tels que définis dans la description. Les complexes de palladium sont utiles dans des procédés de fluoration de substrats aryle et hétéroaryle. La présente invention concerne également des compositions et des kits comprenant lesdits complexes de palladium.
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)