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1. (WO2017134588) PROCESS FOR THE PREPARATION OF IBRUTINIB
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2017/134588 International Application No.: PCT/IB2017/050553
Publication Date: 10.08.2017 International Filing Date: 02.02.2017
IPC:
C07D 487/04 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
487
Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/-C07D477/183
02
in which the condensed system contains two hetero rings
04
Ortho-condensed systems
Applicants:
SHILPA MEDICARE LIMITED [IN/IN]; #12-6-214/A1, Hyderabad Road, Karnataka Raichur 584135, IN
Inventors:
RAMPALLI, Sriram; IN
UPALLA, Lav Kumar; IN
PATNEEDI, Chanti Babu; IN
DASARI, Gopala Krishna; IN
CHATURVEDI, Akshay Kant; IN
Priority Data:
20164100408004.02.2016IN
Title (EN) PROCESS FOR THE PREPARATION OF IBRUTINIB
(FR) PROCÉDÉ DE PRÉPARATION D'IBRUTINIB
Abstract:
(EN) The present invention relates to a process for the preparation of 1-[(3R)-3 -[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl] -1-piperidinyl]-2-propen-1-one or Ibrutinib of Formula (I). The present invention further relates to a process for the preparation highly pure 1-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)-1 H-pyrazolo[3,4-d]pyrimidin-1-yl] -1-piperidinyl]-2-propen-l-one or Ibrutinib.
(FR) La présente invention concerne un procédé de préparation de 1-[(3R)-3-[4-amino-3-(4-phénoxyphényl)-1H-pyrazolo [3,4-d] pyrimidin-1-yl]-1-pipéridinyl]-2-propen-1-one ou ibrutinib de Formule (I). L'invention concerne également un procédé de préparation de 1-[(3R)-3-[4-amino-3-(4-phénoxyphényl)-1H-pyrazolo [3,4-d] pyrimidin-1-yl]-1-pipéridinyl]-2-propen-1-one ou ibrutinib (I) de grande pureté.
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)
Also published as:
US20190040069