Search International and National Patent Collections
Some content of this application is unavailable at the moment.
If this situation persists, please contact us atFeedback&Contact
1. (WO2017134087) STEROIDIC CALIXARENE COMPOUNDS, THEIR SYNTHESIS AND USE FOR EXTRACTION, SOLUBILIZATION AND/OR STABILIZATION OF NATIVE AND FUNCTIONAL MEMBRANE PROTEINS
Latest bibliographic data on file with the International Bureau

Pub. No.: WO/2017/134087 International Application No.: PCT/EP2017/052118
Publication Date: 10.08.2017 International Filing Date: 01.02.2017
IPC:
C07J 9/00 (2006.01) ,C07J 43/00 (2006.01) ,C07J 71/00 (2006.01) ,C07K 1/14 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
J
STEROIDS
9
Normal steroids containing carbon, hydrogen, halogen, or oxygen, substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
J
STEROIDS
43
Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta[a]hydrophenanthrene skeleton
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
J
STEROIDS
71
Steroids in which the cyclopenta[a]hydrophenanthrene skeleton is condensed with a heterocyclic ring
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
K
PEPTIDES
1
General processes for the preparation of peptides
14
Extraction; Separation; Purification
Applicants:
CALIXAR [FR/FR]; 60 avenue Rockefeller 69008 Lyon, FR
Inventors:
DAUVERGNE, Julien; FR
JAWHARI, Anass; FR
LESSAULT, Morgane; FR
OURRI, Benjamin; FR
Agent:
SCHMIDT, Martin; FR
Priority Data:
1601895.403.02.2016GB
Title (EN) STEROIDIC CALIXARENE COMPOUNDS, THEIR SYNTHESIS AND USE FOR EXTRACTION, SOLUBILIZATION AND/OR STABILIZATION OF NATIVE AND FUNCTIONAL MEMBRANE PROTEINS
(FR) COMPOSÉS STÉROÏDIQUES DE CALIXARÈNE, LEUR SYNTHÈSE ET LEUR UTILISATION POUR L'EXTRACTION, LA SOLUBILISATION ET/OU LA STABILISATION DE PROTÉINES MEMBRANAIRES NATIVES ET FONCTIONNELLES
Abstract:
(EN) Steroidic calixarene compounds according to formula (I): (I) wherein: ∙ R represents -(CH2)x-L-(CH2)y-Ster, wherein : ○ x and y are integers comprised between 0 and 2; ○ n is an integer comprised between 1 and 5; ○ L represents an oxygen atom, an amide spacer –NHCO-, a 1,2,3-triazole spacer, or can be absent; ○ Ster represents a structure derived from a steroid. ∙ X represents H or Y, wherein: ○ Y represents -(CH2)m-CO2Z wherein m is an integer comprised between 0 and 2; ○ Z represents an alkali metal.
(FR) L'invention concerne des composés stéroïdiques de calixarène de formule (I) : (I) où : ∙ R représente (CH2)x-L-(CH2)y-Ster, où : ○ x et y sont des nombres entiers compris entre 0 et 2 ; ○ n est un nombre entier compris entre 1 et 5 ; ○ L représente un atome d'oxygène, un espaceur amide –NHCO-, un espaceur 1,2,3-triazole, ou il peut être absent ; ○ Ster représente une structure dérivée d'un stéroïde. ∙ X représente H ou Y, où : ○ Y représente (CH2)m-CO2Z où m est un nombre entier compris entre 0 et 2 ; ○ Z représente un métal alcalin.
front page image
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)