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1. (WO2017066428) BRD4-KINASE INHIBITORS AS CANCER THERAPEUTICS
Latest bibliographic data on file with the International Bureau    Submit observation

Pub. No.: WO/2017/066428 International Application No.: PCT/US2016/056811
Publication Date: 20.04.2017 International Filing Date: 13.10.2016
IPC:
A61K 31/506 (2006.01) ,C07D 239/48 (2006.01)
Applicants: H. LEE MOFFITT CANCER CENTER & RESEARCH INSTITUTE, INC.[US/US]; 12902 Magnolia Drive Tampa, Florida 33612-9497, US
Inventors: SCHÖNBRUNN, Ernst; US
LAWRENCE, Nicholas J.; US
LAWRENCE, Harshani R.; US
Agent: CURFMAN, Christopher L.; US
HALL, Miles E.; US
GILES, P. Brian; US
Priority Data:
62/240,87113.10.2015US
Title (EN) BRD4-KINASE INHIBITORS AS CANCER THERAPEUTICS
(FR) INHIBITEURS DE BRD4-KINASE À UTILISER EN TANT QU'AGENTS THÉRAPEUTIQUES ANTICANCÉREUX
Abstract: front page image
(EN) Disclosed herein are compounds that are inhibitors of BDR4 and their use in the treatment of cancer. Methods of screening for selective inhibitors of BDR4 are also disclosed. In certain aspects, disclosed are compounds of Formula I through IV.
(FR) La présente invention concerne des composés qui sont des inhibiteurs de BRD4 et leur utilisation dans le traitement du cancer. L'invention concerne également des procédés de criblage d'inhibiteurs sélectifs de BDR4. Dans certains aspects, l'invention concerne des composés de formule I-IV.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)