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1. (WO2017036266) 3-ARYL PYRIDAZINONE, PREPARATION METHOD, PESTICIDE COMPOSITION AND USE
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2017/036266 International Application No.: PCT/CN2016/092002
Publication Date: 09.03.2017 International Filing Date: 28.07.2016
IPC:
C07D 237/14 (2006.01) ,C07D 417/04 (2006.01) ,C07D 413/04 (2006.01) ,A01N 43/58 (2006.01) ,A01N 43/76 (2006.01) ,A01N 43/78 (2006.01) ,A01N 43/84 (2006.01) ,A01P 13/00 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
237
Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
02
not condensed with other rings
06
having three double bonds between ring members or between ring members and non-ring members
10
with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
14
Oxygen atoms
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
417
Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/196
02
containing two hetero rings
04
directly linked by a ring-member-to-ring- member bond
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
413
Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
02
containing two hetero rings
04
directly linked by a ring-member-to-ring- member bond
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
N
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43
Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
48
having rings with two nitrogen atoms as the only ring hetero atoms
58
1,2-Diazines; Hydrogenated 1,2-diazines
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
N
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43
Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
72
having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms
74
five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
76
1,3-Oxazoles; Hydrogenated 1,3-oxazoles
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
N
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43
Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
72
having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms
74
five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
78
1,3-Thiazoles; Hydrogenated 1,3-thiazoles
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
N
PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
43
Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
72
having rings with nitrogen atoms and oxygen or sulfur atoms, as ring hetero atoms
84
six-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,4
A HUMAN NECESSITIES
01
AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
P
BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
13
Herbicides; Algicides
Applicants:
中国科学院上海有机化学研究所 SHANGHAI INSITITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES [CN/CN]; 中国上海市 徐汇区零陵路345号 No.345, Lingling Road, Xuhui District Shanghai 200032, CN
Inventors:
吕龙 LV, Long; CN
吕强 LV, Qiang; CN
唐庆红 TANG, Qinghong; CN
付群梅 FU, Qunmei; CN
张基胜 ZHANG, Jisheng; CN
刘世梦 LIU, Shimeng; CN
戴明 DAI, Ming; CN
张志国 ZHANG, Zhiguo; CN
沈娟 SHEN, Juan; CN
芦昕婷 LU, Xinting; CN
Agent:
上海弼兴律师事务所 SHANGHAI BESHINING LAW OFFICE; 中国上海市 小木桥路681号外经大厦21楼 21st Floor, SFECO Mansion, No.681 Xiaomuqiao Road Shanghai 200032, CN
Priority Data:
201510559286.102.09.2015CN
Title (EN) 3-ARYL PYRIDAZINONE, PREPARATION METHOD, PESTICIDE COMPOSITION AND USE
(FR) 3-ARYL PYRIDAZINONE, PROCÉDÉ DE PRÉPARATION, COMPOSITION PESTICIDE ET UTILISATION
(ZH) 3-芳基哒嗪酮类化合物、制备方法、农药组合物及用途
Abstract:
(EN) Provided are 3-aryl pyridazinone as shown by formula I, and a preparation method, pesticide composition and use. The 3-aryl pyridazinone provided has a highly-efficient herbicidal activity, a relatively broad phytocidal range, good crop safety, a relatively wide drug application period, and a short residual life in the soil; the 3-aryl pyridazinone exhibits good pre-emergence and post-emergence herbicidal activity at low doses, has control effects on all of farmland broadleaved weeds, farmland gramineae weeds and Cyperaceae weeds, and has a certain safety for crops such as corn, rice, wheat, cotton and soybeans at high doses; the 3-aryl pyridazinone can effectively inhibit the germination of weeds, and at the same time has a good herbicidal activity on 3-6 leaf-stage sensitive large weeds and no harmful effects on the growth of succeeding crops; and the 3-aryl pyridazinone has a reasonable toxicity, ecotoxicity and environmental capability, belonging to environmentally friendly low-toxic pesticides with good market prospects.
(FR) La présente invention concerne une 3-aryl pyridazinone telle que présentée par la formule I, et un procédé de préparation, une composition pesticide et une utilisation. La 3-aryl pyridazinone décrite possède une activité herbicide hautement efficace, une plage phytocide relativement large, une bonne innocuité vis-à-vis des cultures, une période d’application du médicament relativement large, et une courte durée de vie résiduelle dans le sol ; la 3-aryl pyridazinone fait preuve d’une bonne activité herbicide pré-levée et post-levée à faibles doses, possède des effets de régulation sur l’ensemble des mauvaises herbes agricoles à larges feuilles, sur les mauvaises herbes agricoles des graminées et les mauvaises herbes de la famille des Cyperaceae, et présente une certaine innocuité vis-à-vis des cultures telles que le maïs, le riz, le blé, le coton et le soja à doses élevées ; la 3-aryl pyridazinone peut inhiber de manière efficace la germination des mauvaises herbes, et en même temps présenter une bonne activité herbicide sur les grandes mauvaises herbes sensibles au stade 3 à 6 feuilles et sans effets nuisibles sur le développement des cultures ultérieures ; et la 3-aryl pyridazinone fait preuve d’une toxicité, écotoxicité et capacité environnementale raisonnables, appartenant aux pesticides peu toxiques respectueux de l’environnement ayant de bonnes perspectives commerciales.
(ZH) 提供了一种如式(I)所示的3-芳基哒嗪酮类化合物、制备方法、农药组合物及用途。提供的3-芳基哒嗪酮类化合物具有高效的除草活性、杀草谱较广、作物安全性良好、施药期较宽、土壤中残留期短、在低剂量下表现出良好的芽前和芽后除草活性,对农田阔叶杂草、农田禾本科杂草和莎草科杂草均具有控制效果,高剂量下对玉米、水稻、小麦、棉花、大豆等作物具有一定的安全性,能较好的抑制杂草出芽,同时对大龄3~6叶期敏感杂草也具有良好的除草活性,对后茬作物生长无不良影响,具有合理的毒性、生态毒性和环境相容性,属低毒环境友好型农药,有良好的市场化前景。
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Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: Chinese (ZH)
Filing Language: Chinese (ZH)