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1. WO2016193240 - AMINOESTER DERIVATIVES USEFUL IN THE TREATMENT OF COPD

Publication Number WO/2016/193240
Publication Date 08.12.2016
International Application No. PCT/EP2016/062223
International Filing Date 31.05.2016
IPC
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
401
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
02
containing two hetero rings
12
linked by a chain containing hetero atoms as chain links
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
453
Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
02
containing not further condensed quinuclidine ring systems
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
435
having six-membered rings with one nitrogen as the only ring hetero atom
44
Non-condensed pyridines; Hydrogenated derivatives thereof
445
Non-condensed piperidines, e.g. piperocaine
4523
containing further heterocyclic ring systems
4545
containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
11
Drugs for disorders of the respiratory system
C07D 401/12 (2006.01)
C07D 453/02 (2006.01)
A61K 31/4545 (2006.01)
A61P 11/00 (2006.01)
CPC
A61K 31/444
A61K 31/452
C07D 401/12
C07D 453/02
Applicants
  • CHIESI FARMACEUTICI S.P.A. [IT/IT]; Via Palermo, 26/A 43100 Parma, IT
Inventors
  • AMARI, Gabriele; IT
  • ARMANI, Elisabetta; IT
  • VAN DE PÖEL, Hervé; IT
  • BAKER-GLENN, Charles; IT
  • TRIVEDI, Naimisha; IT
Agents
  • MINOJA, Fabrizio; IT
Priority Data
15170047.301.06.2015EP
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) AMINOESTER DERIVATIVES USEFUL IN THE TREATMENT OF COPD
(FR) DÉRIVÉS D'AMINOESTERS UTILES POUR TRAITER LA BPCO
Abstract
(EN)
The invention relates to novel compounds which are both phosphodiesterase 4 (PDE4) enzyme inhibitors and muscarinic M3 receptor antagonists, methods of preparing such compounds, compositions containing them and therapeutic use thereof.
(FR)
La présente invention concerne de nouveaux composés qui sont à la fois des inhibiteurs d'enzyme phosphodiestérase 4 (PDE4) et des antagonistes des récepteurs muscariniques M3, des procédés de préparation de tels composés, des compositions les contenant et leur utilisation thérapeutique.
Also published as
Latest bibliographic data on file with the International Bureau