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1. WO2016177849 - AMINOESTER DERIVATIVES

Publication Number WO/2016/177849
Publication Date 10.11.2016
International Application No. PCT/EP2016/060122
International Filing Date 05.05.2016
IPC
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
409
Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
02
containing two hetero rings
12
linked by a chain containing hetero atoms as chain links
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
409
Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
14
containing three or more hetero rings
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
D
HETEROCYCLIC COMPOUNDS
471
Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/-C07D463/251
02
in which the condensed system contains two hetero rings
08
Bridged systems
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
435
having six-membered rings with one nitrogen as the only ring hetero atom
439
the ring forming part of a bridged ring system, e.g. quinuclidine
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
P
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
11
Drugs for disorders of the respiratory system
C07D 409/12 (2006.01)
C07D 409/14 (2006.01)
C07D 471/08 (2006.01)
A61K 31/439 (2006.01)
A61P 11/00 (2006.01)
CPC
A61K 31/439
A61K 31/4436
A61K 31/4439
A61K 31/4545
C07D 409/12
C07D 409/14
Applicants
  • CHIESI FARMACEUTICI S.P.A. [IT/IT]; Via Palermo, 26/A 43100 Parma, IT
Inventors
  • AMARI, Gabriele; IT
  • ARMANI, Elisabetta; IT
  • BLACKABY, Wesley; IT
  • VAN DE PÖEL, Hervé; IT
  • BAKER-GLENN, Charles; IT
  • TRIVEDI, Naimisha; IT
Agents
  • MINOJA, Fabrizio; IT
Priority Data
15166703.707.05.2015EP
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) AMINOESTER DERIVATIVES
(FR) DÉRIVÉS D'AMINOESTERS
Abstract
(EN)
The invention relates to novel compounds which are both phosphodiesterase 4 (PDE4) enzyme inhibitors and muscarinic M3 receptor antagonists, methods of preparing such compounds, compositions containing them and therapeutic use thereof.
(FR)
L'invention concerne de nouveaux composés qui sont à la fois des inhibiteurs de l'enzyme phosphodiestérase 4 (PDE4) et des antagonistes des récepteurs muscariniques M3, des procédés de préparation de tels composés, des compositions les contenant et leur utilisation thérapeutique.
Also published as
Latest bibliographic data on file with the International Bureau