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1. (WO2016105529) METHODS FOR PREPARING FUSED BICYCLIC 2, 4-DIAMINOPYRIMIDINE DERIVATIVES
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2016/105529    International Application No.:    PCT/US2015/000301
Publication Date: 30.06.2016 International Filing Date: 23.12.2015
IPC:
C07D 403/12 (2006.01), C07D 295/135 (2006.01)
Applicants: CEPHALON, INC. [US/US]; 41 Moores Road PO Box 4011 Frazer, PA 19355 (US)
Inventors: ALLWEIN, Shawn, P.; (US).
BAKALE, Roger, P.; (US).
MOWREY, Dale, R.; (US).
PETRILLO, Daniel, E.; (US).
KLUWER, Sander; (NL)
Agent: VALLA, S, Maurice; (US)
Priority Data:
62/095,861 23.12.2014 US
Title (EN) METHODS FOR PREPARING FUSED BICYCLIC 2, 4-DIAMINOPYRIMIDINE DERIVATIVES
(FR) PROCÉDÉS DE PRÉPARATION DE DÉRIVÉS DE 2, 4-DIAMINOPYRIMIDINE BICYCLIQUES FUSIONNÉS
Abstract: front page image
(EN)The present disclosure is directed to improved methods useful for the preparation of, for example, 2-[[5-chloro-2-[[(6S)-6-[4-(2-hydroxyethyl)piperazin-l-yl]-l-methoxy-6,7,8,9- tetrahydro-5Hbenzo[7]annulen-2-yl]amino]pyrimidin-4-yl]amino]-N-methyl-benzamide (CEP- 37440).
(FR)La présente invention concerne des procédés améliorés utiles par exemple pour la préparation de 2-[[5-chloro-2-[[(6S)-6-[4-(2-hydroxyéthyl)pipérazin-l-yl]-l-méthoxy-6,7,8,9-tétrahydro-5Hbenzo[7]annulén-2-yl]amino]pyrimidin-4-yl]amino]-N-méthyl-benzamide (CEP-37440).
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)