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1. (WO2016105453) SOLID FORMS OF AN ASK1 INHIBITOR
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2016/105453    International Application No.:    PCT/US2015/000162
Publication Date: 30.06.2016 International Filing Date: 22.12.2015
IPC:
C07D 401/14 (2006.01), C07D 413/12 (2006.01), A61P 3/00 (2006.01), A61P 13/12 (2006.01), A61P 1/16 (2006.01), A61K 31/42 (2006.01), A61K 31/44 (2006.01)
Applicants: GILEAD SCIENCES, INC. [US/US]; 333 Lakeside Drive Foster City, CA 94404 (US)
Inventors: ANDRES, Mark; (US).
CARRA, Ernest, A.; (US).
CHAN, Brenda, J. Burke; (US).
CHIU, Anna; (US).
LAPINA, Olga, Viktorovna; (US).
LATHROP, Stephen, P.; (US).
SMOLENSKAYA, Valeriya; (US).
YU, Lok, Him; (US).
NOTTE, Gregory; (US)
Agent: TANNER, Lorna, L.; (US)
Priority Data:
62/269,066 17.12.2015 US
62/096,406 23.12.2014 US
Title (EN) SOLID FORMS OF AN ASK1 INHIBITOR
(FR) FORMES SOLIDES D'UN INHIBITEUR D'ASK 1
Abstract: front page image
(EN)Crystalline forms of 5-(4-cyclopropyl-1H-imidazol-1-yl)-N-(6-(4-isopropyl-4H-1,2,4-triazol-3-yl)pyridin-2-yl)-2-fluoro-4-methylbenzamide (Compound I) were prepared and characterized in the solid state: Also provided are processes of manufacture and methods of using the crystalline forms.
(FR)La présente invention concerne des formes cristallines de 5-(4-cyclopropyl -1H-imidazol-1-yl)-N-(6-(4-isopropyl-4 H-1,2,4-triazol-3-yl) pyridin-2-yl)-2-fluoro-4-méthylbenzamide (composé I) préparées et caractérisées à l'état solide : L'invention concerne également des procédés de fabrication et des procédés d'utilisation des formes cristallines.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)