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1. (WO2016096140) PROCESS FOR THE PREPARATION OF 1-[(HETEROARYL)-METHYL]- OR 1-[(ARYL)-METHYL]-3-[4-(HYDROXYMETHYL)-PHENYL]-UREAS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2016/096140    International Application No.:    PCT/EP2015/002552
Publication Date: 23.06.2016 International Filing Date: 18.12.2015
IPC:
C07D 231/12 (2006.01), A61K 31/415 (2006.01), A61P 29/00 (2006.01)
Applicants: GRÜNENTHAL GMBH [DE/DE]; Zieglerstrasse 6 52078 Aachen (DE)
Inventors: WESQUET, Alexander; (DE).
WITTLAND, Claudia; (DE).
GRIEBEL, Carsten; (DE).
ZIMMER, Oswald; (DE)
Priority Data:
14004300.1 19.12.2014 EP
Title (EN) PROCESS FOR THE PREPARATION OF 1-[(HETEROARYL)-METHYL]- OR 1-[(ARYL)-METHYL]-3-[4-(HYDROXYMETHYL)-PHENYL]-UREAS
(FR) PROCÉDÉ POUR LA PRÉPARATION DE 1-[(HÉTÉROARYL)-MÉTHYL] OU 1- [(ARYL)-MÉTHYL] -3- [4-(HYDROXYMÉTHYL)-PHÉNYL]-URÉES
Abstract: front page image
(EN)The present invention relates to a process for the preparation of certain 1-[(heteroaryl)-methyl]-3-[4- (hydroxymethyl)-phenyl]-ureas or 1-[(aryl)-methyl]-3-[4-(hydroxymethyl)-phenyl]-ureas, in particular certain 1-[(2-aryl-2H-pyrazol-3-yl)-methyl]-3-[4-(hydroxymethyl)-phenyl]-ureas or physiologically acceptable addition salts and/or solvates thereof.
(FR)La présente invention concerne un procédé pour la préparation de certaines 1-[(hétéroaryl)-méthyl]-3-[4- (hydroxyméthyl)-phényl]-urées ou 1-[(aryle)-méthyl]-3- [4-(hydroxyméthyl)-phényl]-urées, en particulier certaines 1-[(2-aryl-2H-pyrazol-3-yl)-méthyl]-3-[4- (hydroxyméthyl)-phényl]-urées ou des sels d'addition et/ou solvates physiologiquement acceptables associés.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)