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1. (WO2016092375) SUBSTITUTED HETEROCYCLES AS BROMODOMAIN INHIBITORS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2016/092375    International Application No.:    PCT/IB2015/002479
Publication Date: 16.06.2016 International Filing Date: 11.12.2015
IPC:
C07D 403/14 (2006.01), A61K 31/4196 (2006.01), A61K 31/4439 (2006.01), A61K 31/4985 (2006.01), C07D 401/14 (2006.01), C07D 403/04 (2006.01), C07D 413/14 (2006.01)
Applicants: ZENITH EPIGENETICS LTD. [CA/CA]; 300, 4820 Richard Road SW Calgary. AB, T3E 6L1 (CA)
Inventors: BROWN, Samuel, David; (US).
COBURN, Craig, Alan; (US).
KHARENKO, Olesya; (CA)
Priority Data:
62/090,853 11.12.2014 US
Title (EN) SUBSTITUTED HETEROCYCLES AS BROMODOMAIN INHIBITORS
(FR) HÉTÉROCYCLES SUBSTITUÉS À TITRE D'INHIBITEURS DE BROMODOMAINES
Abstract: front page image
(EN)The present application relates to substituted heterocycles compound of Formula I and pharmaceutical compositions thereof useful for the inhibition of BET protein function by binding to bromodomains (Formula I).
(FR)Cette invention concerne des composés hétérocycles substitués de Formule I et des compositions pharmaceutiques les contenant utiles pour inhiber la fonction protéique BET par liaison des bromodomaines (Formule I).
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)