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1. (WO2016055644) LINEAR GUANIDINE DERIVATIVES, METHODS OF PREPARATION AND USES THEREOF

Pub. No.:    WO/2016/055644    International Application No.:    PCT/EP2015/073467
Publication Date: Fri Apr 15 01:59:59 CEST 2016 International Filing Date: Sat Oct 10 01:59:59 CEST 2015
IPC: A61K 31/155
C07C 279/04
C08K 5/31
Applicants: LEAD DISCOVERY SIENA S.R.L.
Inventors: BOTTA, Maurizio
MACCARI, Giorgio
SANFILIPPO, Stefania
DE LUCA, Filomena
DOCQUIER, Jean-Denis
DEODATO, Davide
Title: LINEAR GUANIDINE DERIVATIVES, METHODS OF PREPARATION AND USES THEREOF
Abstract:
The present invention relates to linear guanidine derivatives, methods of preparation, uses and pharmaceutical compositions thereof. The compounds of Formulas 1 or 2 exhibit high antimicrobial activity against Gram positive and Gram negative bacteria.