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Machine translation
1. (WO2014195593) ACETYLCHOLINESTERASE INHIBITOR COMPOUNDS AND 5HT4 SEROTONERGIC RECEPTOR AGONISTS, WITH PROMNESIA EFFECT, METHODS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2014/195593    International Application No.:    PCT/FR2014/051149
Publication Date: 11.12.2014 International Filing Date: 19.05.2014
IPC:
C07D 211/20 (2006.01), A61K 31/445 (2006.01), C07D 211/26 (2006.01), C07D 211/32 (2006.01), A61P 25/28 (2006.01)
Applicants: UNIVERSITE DE CAEN [FR/FR]; Esplanade de la Paix F-14000 Caen (FR)
Inventors: DALLEMAGNE, Patrick; (FR).
ROCHAIS, Christophe; (FR).
LECOUTEY, Cédric; (FR).
BOULOUARD, Michel; (FR).
FRERET, Thomas; (FR)
Agent: CABINET MALEMONT; 91 avenue Kléber F-75116 Paris (FR)
Priority Data:
1355155 05.06.2013 FR
Title (EN) ACETYLCHOLINESTERASE INHIBITOR COMPOUNDS AND 5HT4 SEROTONERGIC RECEPTOR AGONISTS, WITH PROMNESIA EFFECT, METHODS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
(FR) COMPOSES INHIBITEURS DE L'ACETYLCHOLINESTERASE ET AGONISTES DES RECEPTEURS SEROTONINERGIQUES 5HT4, A EFFET PROMNESIANT, LEURS PROCEDES DE PREPARATION ET COMPOSITIONS PHARMACEUTIQUES LES CONTENANT
Abstract: front page image
(EN)The invention relates to compounds of formula (I) as well as to neurogenic enantiomers thereof, acid salts thereof, hydrates thereof or to solvation products thereof. Among a large number of possible meanings, X is a halogen, Y is an oxygen atom; all the coefficients m, n, r and s have a value of 1, R is a methyl, and R' is a cycloalkyl. The invention also includes methods for preparing the above compounds and pharmaceutical compositions including same.
(FR)L'invention concerne des composés de formule (I) ainsi que leur énantiomères neurocéniques, leurs sels d'acide, leurs hydrates ou leurs produits de solvatation. Parmi un grand nombre de significations possible, X représente un halogène, Y un atome d'oxygène; tous les coefficients m,n,r et s ont la valeur 1, R représente un méthyl et R' un cycloalkyl. L'invention comprend également des procédés de préparation des composés ci-dessus et des compositions pharmaceutiques les comprenant.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG).
Publication Language: French (FR)
Filing Language: French (FR)