Some content of this application is unavailable at the moment.
If this situation persist, please contact us atFeedback&Contact
1. (WO2014193837) SYNTHESIS OF GALANAL COMPOUNDS AND ANALOGUES THEREOF
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2014/193837 International Application No.: PCT/US2014/039575
Publication Date: 04.12.2014 International Filing Date: 27.05.2014
IPC:
C07C 45/27 (2006.01) ,C07C 47/43 (2006.01) ,C07C 49/413 (2006.01)
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
45
Preparation of compounds having CO groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
27
by oxidation
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
47
Compounds having -CHO groups
38
Unsaturated compounds having -CHO groups bound to carbon atoms of rings other than six-membered aromatic rings
43
with a seven- to twelve-membered ring
C CHEMISTRY; METALLURGY
07
ORGANIC CHEMISTRY
C
ACYCLIC OR CARBOCYCLIC COMPOUNDS
49
Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
385
Saturated compounds containing a keto group being part of a ring
413
of a seven- to twelve-membered ring
Applicants:
ACADEMIA SINICA; 128 Academia Road Section 2, Nankang Taipei, 115, TW
LIANG, Chi-Ming [US/US]; US
Inventors:
KING, Klim; TW
CHEIN, Rong-Jie; TW
Agent:
CHEN, Yahua; Wolf, Greenfield & Sacks, P.C. 600 Atlantic Avenue Boston, MA 02210-2206, US
Priority Data:
61/827,67427.05.2013US
61/839,87027.06.2013US
Title (EN) SYNTHESIS OF GALANAL COMPOUNDS AND ANALOGUES THEREOF
(FR) SYNTHÈSE DE COMPOSÉS DE GALANAL ET LEURS ANALOGUES
Abstract:
(EN) The present disclosure provides methods of preparing glucagon-like peptide-1 (GLP-1) receptor modulators, such as compounds of Formula (II) or (VI), or intermediates thereof. The compounds that may be prepared by the described methods are useful for regulating blood glucose levels and/or treating a disease mediated by a GLP-1 receptor (e.g.diabetes).
(FR) La présente invention concerne des procédés de préparation de modulateurs du récepteur du glucagon-like peptide-1 (GLP-1), tels que des composés de formule (II) ou (VI) ou leurs intermédiaires. Les composés qui peuvent être préparés par les procédés décrits sont utiles dans la régulation des taux de glycémie et/ou le traitement d'une maladie induite par un récepteur de GLP-1 (telle que le diabète).
front page image
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JP, KE, KG, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, KM, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)