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1. WO2013159736 - MONOFLUORO CYCLOPROPANE COMPOUND, AND PREPARATION METHOD AND USE THEREOF

Publication Number WO/2013/159736
Publication Date 31.10.2013
International Application No. PCT/CN2013/074804
International Filing Date 26.04.2013
IPC
C07C 49/327 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
49Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
29Saturated compounds containing keto groups bound to rings
327containing halogen
C07C 49/567 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
49Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
527Unsaturated compounds containing keto groups bound to rings other than six-membered aromatic rings
567containing halogen
C07C 233/59 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
233Carboxylic acid amides
57having carbon atoms of carboxamide groups bound to carbon atoms of rings other than six-membered aromatic rings
59having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups
C07C 259/08 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
259Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
04without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids
08having carbon atoms of hydroxamic groups bound to carbon atoms of rings other than six-membered aromatic rings
C07C 381/10 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
381Compounds containing carbon and sulfur and having functional groups not covered by groups C07C301/-C07C337/142
10Compounds containing sulfur atoms doubly-bound to nitrogen atoms
C07C 35/48 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
35Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring
48Halogenated derivatives
CPC
C07C 259/08
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
259Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
04without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids
08having carbon atoms of hydroxamic groups bound to carbon atoms of rings other than six-membered aromatic rings
C07C 2601/02
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
2601Systems containing only non-condensed rings
02with a three-membered ring
C07C 381/10
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
381Compounds containing carbon and sulfur and having functional groups not covered by groups C07C301/00 - C07C337/00
10Compounds containing sulfur atoms doubly-bound to nitrogen atoms
C07C 43/23
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
43Ethers; Compounds having groups, groups or groups
02Ethers
20having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring
23containing hydroxy or O-metal groups
C07C 47/353
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
47Compounds having —CHO groups
28Saturated compounds having —CHO groups bound to carbon atoms of rings other than six—membered aromatic rings
353containing halogen
C07C 47/457
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
CACYCLIC OR CARBOCYCLIC COMPOUNDS
47Compounds having —CHO groups
38Unsaturated compounds having —CHO groups bound to carbon atoms of rings other than six—membered aromatic rings
457containing halogen
Applicants
  • 中国科学院上海有机化学研究所 SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES [CN]/[CN]
Inventors
  • 胡金波 HU, Jinbo
  • 沈晓 SHEN, Xiao
Agents
  • 上海一平知识产权代理有限公司 XU & PARTNERS, LLC.
Priority Data
201210129611.727.04.2012CN
Publication Language Chinese (ZH)
Filing Language Chinese (ZH)
Designated States
Title
(EN) MONOFLUORO CYCLOPROPANE COMPOUND, AND PREPARATION METHOD AND USE THEREOF
(FR) COMPOSÉ DE CYCLOPROPANE MONOFLUORÉ, ET SON PROCÉDÉ DE PRÉPARATION ET SON UTILISATION
(ZH) 单氟代环丙烷类化合物及其制备方法和应用
Abstract
(EN)
Disclosed are a monofluoro cyclopropane compound, and preparation method and uses thereof. The structure of the monofluoro cyclopropane compound is as represented by formula I, wherein R1, R2, Ra, and formula II are as defined in the specification. Also provided is a method for simply and effectively preparing the monofluoro cyclopropane compound. The method can prepare both racemic compounds and non-racemic compounds. The monofluoro cyclopropane compound can be further used to synthesize other cyclopropane derivatives.
(FR)
La présente invention concerne un composé de cyclopropane monofluoré, et son procédé de préparation et son utilisation. La structure du composé de cyclopropane monofluoré est telle que représentée par la formule I, dans laquelle R1, R2, Ra, et la formule II sont tels que définis dans la description. L'invention concerne également un procédé pour la préparation simple et efficace du composé de cyclopropane monofluoré. Le procédé permet de préparer des composés racémiques ainsi que des composés non racémiques. Le composé de cyclopropane monofluoré peut être également utilisé pour la synthèse d'autres dérivés de cyclopropane.
(ZH)
公开了一种单氟代环丙烷类化合物及其制备方法和应用。单氟代环丙烷类化合物的结构如式I所示,式中,R1,R2,Ra,式II的定义如说明书中所述。还提供了一种简单有效的制备单氟代环丙烷类化合物的方法。该方法不仅能制备消旋的化合物,还可制备非消旋的化合物。单氟代环丙烷类化合物可进一步用于合成其他环丙烷衍生物。
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