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1. (WO2013152741) 4-SUBSTITUENT-2-HYDROXYLMORPHOLINE-3-ONE AND PREPARATION METHOD THEREOF
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2013/152741    International Application No.:    PCT/CN2013/074202
Publication Date: 17.10.2013 International Filing Date: 15.04.2013
IPC:
C07D 265/32 (2006.01), C07D 413/06 (2006.01)
Applicants: ZHEJIANG HISUN PHARMACEUTICAL CO., LTD. [CN/CN]; No.46 Waisha Road, Jiaojiang District Taizhou, Zhejiang 318000 (CN).
SHANGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY [CN/CN]; No.1320 West Beijing Road, Jing'an District Shanghai 200040 (CN)
Inventors: ZHANG, Fuli; (CN).
LIU, Chonghao; (CN).
QIU, Pengcheng; (CN).
CHAI, Jian; (CN).
CAI, Qingfeng; (CN)
Agent: UNITALEN ATTORNEYS AT LAW; 7th Floor, Scitech Place No.22, Jian Guo Men Wai Ave., Chao Yang District Beijing 100004 (CN)
Priority Data:
201210112140.9 13.04.2012 CN
Title (EN) 4-SUBSTITUENT-2-HYDROXYLMORPHOLINE-3-ONE AND PREPARATION METHOD THEREOF
(FR) 2-HYDROXYMORPHOLINE-3-ONE 4-SUBSTITUÉE ET SON PROCÉDÉ DE PRÉPARATION
(ZH) 4-取代基-2-羟基吗啉-3-酮及其制备方法
Abstract: front page image
(EN)A molecule with neuro activities, especially 4-substituent-2-hydroxylmorpholine-3-one, as a new intermediate of neurokinin-1 receptor antagonist Aprepitant, and preparation method thereof.
(FR)Cette invention concerne une molécule ayant des activités neurologiques, notamment la 2-hydroxymorpholine-3-one 4-substituée, à titre de nouvel intermédiaire d'antagoniste du récepteur de neurokinine-1. Un aprépitant, et son procédé de préparation sont également décrits.
(ZH)一类具有神经活性作用的分子,尤其是神经激肽-1受体拮抗剂阿瑞吡坦的新中间体4-取代基-2-羟基吗啉-3-酮及其制备方法。
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: Chinese (ZH)
Filing Language: Chinese (ZH)