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1. (WO2013149136) ISOXAZOLE β-LACTAMASE INHIBITORS
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2013/149136    International Application No.:    PCT/US2013/034589
Publication Date: 03.10.2013 International Filing Date: 29.03.2013
IPC:
C07D 451/06 (2006.01), A61K 31/46 (2006.01), A61P 31/00 (2006.01)
Applicants: CUBIST PHARMACEUTICALS, INC. [US/US]; 65 Hayden Ave Lexington, MA 02421 (US)
Inventors: GU, Yu Gui; (US).
HE, Yong; (US).
YIN, Ning; (US).
ALEXANDER, Dylan, C.; (US).
CROSS, Jason, B.; (US).
METCALF, Chester, A., III.; (US).
BUSCH, Robert; (US)
Agent: TRINQUE, Brian, C.; Lathrop & Gage LLP 28 State Street, Suite 0700 Boston, MA 02109 (US)
Priority Data:
61/790,248 15.03.2013 US
61/618,127 30.03.2012 US
Title (EN) ISOXAZOLE β-LACTAMASE INHIBITORS
(FR) INHIBITEURS DES Β-LACTAMASES DÉRIVÉS D'ISOXAZOLE
Abstract: front page image
(EN)β-Lactamase inhibitor compounds (BLIs) are disclosed, including compounds that have activity against class A, class C or class D β-lactamases. Methods of manufacturing the BLIs, and uses of the compounds in the preparation of pharmaceutical compositions and antibacterial applications are also disclosed.
(FR)L'invention concerne des composés inhibiteurs des β-lactamases (BLI) comprenant des composés ayant une activité contre les β-lactamases de classe A, C ou D. Des procédés de fabrication de BLI, les utilisations des composés dans la préparation de compositions pharmaceutiques et des applications antibactériennes sont également divulgués.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)