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1. (WO2013148227) INSULIN-LIKE GROWTH FACTOR-1 RECEPTOR INHIBITORS
Latest bibliographic data on file with the International Bureau   

Pub. No.: WO/2013/148227 International Application No.: PCT/US2013/031155
Publication Date: 03.10.2013 International Filing Date: 14.03.2013
IPC:
A61K 31/497 (2006.01)
A HUMAN NECESSITIES
61
MEDICAL OR VETERINARY SCIENCE; HYGIENE
K
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31
Medicinal preparations containing organic active ingredients
33
Heterocyclic compounds
395
having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
495
having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
4965
Non-condensed pyrazines
497
containing further heterocyclic rings
Applicants: ROYCHOWDHURY, Abhijit[IN/IN]; IN (US)
SHARMA, Rajiv[US/IN]; IN (US)
MASCARENHAS, Malcolm[IN/IN]; IN (US)
B-RAO, Chandrika[IN/IN]; IN (US)
PATIL, Shashikant, M.[IN/IN]; IN (US)
CHAVAN, Sambhaji[IN/IN]; IN (US)
LAD, Nitin[IN/IN]; IN (US)
KHANNA, Smriti[IN/IN]; IN (US)
DINSMORE, Christopher, J.[US/US]; US (US)
MERCK SHARP & DOHME CORP.[US/US]; 126 East Lincoln Avenue Rahway, New Jersey 07065-0907, US
PIRAMAL ENTERPRISES LIMITED[IN/IN]; Piramal Tower, Ganpatrao Kadam Marg Lower Parel Mumbai 400013, IN
Inventors: ROYCHOWDHURY, Abhijit; IN
SHARMA, Rajiv; IN
MASCARENHAS, Malcolm; IN
B-RAO, Chandrika; IN
PATIL, Shashikant, M.; IN
CHAVAN, Sambhaji; IN
LAD, Nitin; IN
KHANNA, Smriti; IN
DINSMORE, Christopher, J.; US
Common
Representative:
MERCK SHARP & DOHME CORP.; 126 East Lincoln Avenue Rahway, New Jersey 07065-0907, US
Priority Data:
61/616,69128.03.2012US
Title (EN) INSULIN-LIKE GROWTH FACTOR-1 RECEPTOR INHIBITORS
(FR) INHIBITEURS DU RÉCEPTEUR DU FACTEUR 1 DE CROISSANCE ANALOGUE À L'INSULINE
Abstract:
(EN) The present invention relates to compounds that are capable of inhibiting, modulating and/or regulating Insulin-Like-Growth Factor I Receptor and Insulin Receptor. The compounds of the instant invention possess a core structure that comprises a sulfonyl indole moiety. The present invention is also related to the pharmaceutically acceptable salts, hydrates and stereoisomers of these compounds.
(FR) La présente invention concerne des composés qui sont aptes à inhiber, à moduler et/ou à réguler le récepteur du facteur I de croissance analogue à l'insuline et le récepteur de l'insuline. Les composés de la présente invention possèdent une structure cœur qui comprend une fraction sulfonyl indole. La présente invention concerne également des sels, hydrates et stéréoisomères pharmaceutiquement acceptables de ces composés.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW
African Regional Intellectual Property Organization (ARIPO) (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Office (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (EPO) (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG)
Publication Language: English (EN)
Filing Language: English (EN)