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1. (WO2013059146) SOLID DOSAGE FORMS OF (S)-ETHYL 2-AMINO-3-(4-(2-AMINO-6-((R)-1-(4-CHLORO-2-(3-METHYL-1H-PYRAZOL-1-YL)PHENYL)-2,2,2-TRIFLUOROETHOXY)PYRIMIDIN-4-YL)PHENYL)PROPANOATE
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2013/059146    International Application No.:    PCT/US2012/060338
Publication Date: 25.04.2013 International Filing Date: 16.10.2012
IPC:
A61K 9/16 (2006.01), A61K 9/20 (2006.01)
Applicants: LEXICON PHARMACEUTICALS, INC. [US/US]; 8800 Technology Forest Place The Woodlands, TX 77381 (US) (For All Designated States Except US).
CHEN, Jinling [US/US]; (US) (US only).
DEAVER, Matthew S. [US/US]; (US) (US only).
HOLL, Richard J. [US/US]; (US) (US only).
NUGURU, Kalyan [IN/US]; (US) (US only)
Inventors: CHEN, Jinling; (US).
DEAVER, Matthew S.; (US).
HOLL, Richard J.; (US).
NUGURU, Kalyan; (US)
Agent: BACHRACH, Max; Lexicon Pharmaceuticals, Inc. 8800 Technology Forest Place The Woodlands, TX 77381 (US)
Priority Data:
61/547,894 17.10.2011 US
Title (EN) SOLID DOSAGE FORMS OF (S)-ETHYL 2-AMINO-3-(4-(2-AMINO-6-((R)-1-(4-CHLORO-2-(3-METHYL-1H-PYRAZOL-1-YL)PHENYL)-2,2,2-TRIFLUOROETHOXY)PYRIMIDIN-4-YL)PHENYL)PROPANOATE
(FR) FORMES POSOLOGIQUES SOLIDES DE (S)-ÉTHYL 2-AMINO-3-(4-(2-AMINO-6-((R)-1-(4-CHLORO-2-(3-MÉTHYL-1H-PYRAZOL-1-YL)PHÉNYL)-2,2,2-TRIFLUOROÉTHOXY)PYRIMIDIN-4-YL)PHÉNYL)PROPANOATE
Abstract: front page image
(EN)Solid pharmaceutical dosage forms comprising (S)-ethyl 2-amino-3-(4-(2-amino-6-((R)-1-(4-chloro-2-(3-methyl-1H-pyrazol-1-yl)phenyl)-2,2,2-trifluoroethoxy)pyrimidin-4-yl)phenyl)propanoate (telotristat) are disclosed, as well as methods of making them and compositions useful in their manufacture.
(FR)L'invention concerne des formes posologiques pharmaceutiques solides comprenant (S)-éthyl 2-amino-3-(4-(2-amino-6-((R)-1-(4-chloro-2-(3-méthyl-1H-pyrazol-1-yl)phényl)-2,2,2-trifluoroéthoxy)pyrimidin-4-yl)phényl)propanoate (télotristat), ainsi que des procédés de fabrication de ceux-ci et des compositions utilisées dans leur fabrication.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KR, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)