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1. WO2013010679 - SALTS OF AZA-BICYCLIC DI-ARYL ETHERS AND METHODS TO MAKE THEM OR THEIR PRECURSORS

Publication Number WO/2013/010679
Publication Date 24.01.2013
International Application No. PCT/EP2012/050517
International Filing Date 13.01.2012
IPC
C07D 453/02 2006.01
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
453Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
02containing not further condensed quinuclidine ring systems
A61K 31/439 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
435having six-membered rings with one nitrogen as the only ring hetero atom
439the ring forming part of a bridged ring system, e.g. quinuclidine
A61P 25/16 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25Drugs for disorders of the nervous system
14for treating abnormal movements, e.g. chorea, dyskinesia
16Anti-Parkinson drugs
A61P 25/18 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25Drugs for disorders of the nervous system
18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
A61P 25/22 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25Drugs for disorders of the nervous system
22Anxiolytics
A61P 25/24 2006.01
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
25Drugs for disorders of the nervous system
24Antidepressants
CPC
A61K 2300/00
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
2300Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
A61K 31/194
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic, hydroximic acids
19Carboxylic acids, e.g. valproic acid
194having two or more carboxyl groups, e.g. succinic, maleic or phthalic acid
A61K 31/439
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
395having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
435having six-membered rings with one nitrogen as the only ring hetero atom
439the ring forming part of a bridged ring system, e.g. quinuclidine
A61K 9/2054
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
9Medicinal preparations characterised by special physical form
20Pills, tablets, ; discs, rods
2004Excipients; Inactive ingredients
2022Organic macromolecular compounds
205Polysaccharides, e.g. alginate, gums; Cyclodextrin
2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
A61P 15/10
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
15Drugs for genital or sexual disorders
10for impotence
A61P 19/02
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
19Drugs for skeletal disorders
02for joint disorders, e.g. arthritis, arthrosis
Applicants
  • NOVARTIS AG [CH]/[CH] (AllExceptUS)
  • MARTERER, Wolfgang [DE]/[CH] (UsOnly)
  • PRASHAD, Mahavir [US]/[US] (UsOnly)
  • VILLHAUER, Edwin Bernard [US]/[US] (UsOnly)
  • WAYKOLE, Liladhar Murlidhar [US]/[US] (UsOnly)
  • VIVELO, James Anthony [US]/[US] (UsOnly)
  • SUTTER, Bertrand [FR]/[CH] (UsOnly)
  • BIANCHI, Jean-Claude [FR]/[CH] (UsOnly)
  • WU, Raeann [US]/[US] (UsOnly)
  • HAR, Denis [US]/[US] (UsOnly)
  • KARPINSKI, Piotr H. [US]/[US] (UsOnly)
  • PIGNONE, Massimo [IT]/[CH] (UsOnly)
  • STINGELIN, Doris [CH]/[CH] (UsOnly)
  • BUERGER, Eckart [CH]/[CH] (UsOnly)
Inventors
  • MARTERER, Wolfgang
  • PRASHAD, Mahavir
  • VILLHAUER, Edwin Bernard
  • WAYKOLE, Liladhar Murlidhar
  • VIVELO, James Anthony
  • SUTTER, Bertrand
  • BIANCHI, Jean-Claude
  • WU, Raeann
  • HAR, Denis
  • KARPINSKI, Piotr H.
  • PIGNONE, Massimo
  • STINGELIN, Doris
  • BUERGER, Eckart
Agents
  • WIESSNER, Michael
Priority Data
61/508,14715.07.2011US
Publication Language English (EN)
Filing Language English (EN)
Designated States
Title
(EN) SALTS OF AZA-BICYCLIC DI-ARYL ETHERS AND METHODS TO MAKE THEM OR THEIR PRECURSORS
(FR) SELS D'ÉTHERS DIARYLIQUES AZA-BICYCLIQUES ET PROCÉDÉS POUR FABRIQUER CEUX-CI OU LEURS PRÉCURSEURS
Abstract
(EN)
The present invention relates to salts of (R)-3-(6-(4-methylphenyl)-pyridin-3-yloxy)-1-aza- bicyclo[2.2.2]octane, to methods for making them or their precursors, to pharmaceutical compositions comprising them, and to their use as medicaments.
(FR)
La présente invention concerne des sels de (R)-3-(6-(4-méthylphényl)-pyridin-3-yloxy)-1-aza- bicyclo[2.2.2]octane, des procédés pour fabriquer ceux-ci ou leurs précurseurs, des compositions pharmaceutiques comprenant ceux-ci, et leur utilisation en tant que médicaments.
Also published as
Latest bibliographic data on file with the International Bureau