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1. WO2012122264 - OXASPIRO [2.5] OCTANE DERIVATIVES AND ANALOGS

Publication Number WO/2012/122264
Publication Date 13.09.2012
International Application No. PCT/US2012/028068
International Filing Date 07.03.2012
IPC
C07D 303/22 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
303Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
02Compounds containing oxirane rings
12with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
18by etherified hydroxyl radicals
20Ethers with hydroxy compounds containing no oxirane rings
22with monohydroxy compounds
A61K 31/336 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
335having oxygen as the only ring hetero atom, e.g. fungichromin
336having three-membered rings, e.g. oxirane, fumagillin
A61P 3/04 2006.1
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
3Drugs for disorders of the metabolism
04Anorexiants; Antiobesity agents
C07D 303/36 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
303Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
02Compounds containing oxirane rings
36with hydrocarbon radicals, substituted by nitrogen atoms
C07D 303/32 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
303Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
02Compounds containing oxirane rings
12with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
32by aldehydo- or ketonic radicals
C07D 303/34 2006.1
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
303Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
02Compounds containing oxirane rings
34with hydrocarbon radicals, substituted by sulfur, selenium, or tellurium atoms
CPC
A61K 31/336
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
KPREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
31Medicinal preparations containing organic active ingredients
33Heterocyclic compounds
335having oxygen as the only ring hetero atom, e.g. fungichromin
336having three-membered rings, e.g. oxirane, fumagillin
A61P 3/04
AHUMAN NECESSITIES
61MEDICAL OR VETERINARY SCIENCE; HYGIENE
PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
3Drugs for disorders of the metabolism
04Anorexiants; Antiobesity agents
C07B 2200/05
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
2200Indexing scheme relating to specific properties of organic compounds
05Isotopically modified compounds, e.g. labelled
C07B 59/004
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
59Introduction of isotopes of elements into organic compounds ; ; Labelled organic compounds per se
004Acyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium
C07D 303/22
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
303Compounds containing three-membered rings having one oxygen atom as the only ring heteroatom
02Compounds containing oxirane rings
12with hydrocarbon radicals substituted by singly or doubly bound oxygen atoms
18by etherified hydroxyl radicals
20Ethers with hydroxy compounds containing no oxirane rings
22with monohydroxy compounds
C07D 303/32
CCHEMISTRY; METALLURGY
07ORGANIC CHEMISTRY
DHETEROCYCLIC COMPOUNDS
303Compounds containing three-membered rings having one oxygen atom as the only ring heteroatom
02Compounds containing oxirane rings
12with hydrocarbon radicals substituted by singly or doubly bound oxygen atoms
32by aldehydo- or ketonic radicals
Applicants
  • ZAFGEN, INC [US]/[US] (AllExceptUS)
  • VATH, James, E. [US]/[US] (UsOnly)
  • CHAFFEE, Stuart [US]/[US] (UsOnly)
Inventors
  • VATH, James, E.
  • CHAFFEE, Stuart
Agents
  • KAVANAUGH, Theresa, C.
Priority Data
61/450,30108.03.2011US
Publication Language English (en)
Filing Language English (EN)
Designated States
Title
(EN) OXASPIRO [2.5] OCTANE DERIVATIVES AND ANALOGS
(FR) DÉRIVÉS D'OXASPIRO[2.5]OCTANE ET ANALOGUES
Abstract
(EN) The invention provides oxaspiro[2.5]octane derivatives and analogs, methods for preparation thereof, intermediates thereto, pharmaceutical compositions, and uses thereof in the treatment of various disorders and conditions, such as overweight and obesity.
(FR) La présente invention concerne des dérivés et des analogues d'oxaspiro[2.5]octane, leurs procédés de préparation, leurs intermédiaires, des compositions pharmaceutiques et leurs utilisations dans le traitement de divers troubles et diverses pathologies, tels que le surpoids et l'obésité.
Latest bibliographic data on file with the International Bureau