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1. (WO2012115480) DIAMINOPYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2012/115480    International Application No.:    PCT/KR2012/001427
Publication Date: 30.08.2012 International Filing Date: 24.02.2012
IPC:
C07D 403/04 (2006.01), C07D 401/04 (2006.01), A61K 31/506 (2006.01), A61P 1/00 (2006.01)
Applicants: YUHAN CORPORATION [KR/KR]; 49-6 Taebang-dong, Tongjak-gu Seoul 156-754 (KR) (For All Designated States Except US).
LEE, Hyun-Joo [KR/KR]; (KR) (For US Only).
KIM, Dong-Hoon [KR/KR]; (KR) (For US Only).
KIM, Tae-Kyun [KR/KR]; (KR) (For US Only).
YOON, Young-Ae [KR/KR]; (KR) (For US Only).
SIM, Jae-Young [KR/KR]; (KR) (For US Only).
CHA, Myung-Hun [KR/KR]; (KR) (For US Only).
JUNG, Eun-Jung [KR/KR]; (KR) (For US Only).
AHN, Kyoung-Kyu [KR/KR]; (KR) (For US Only).
LEE, Tai-Au [KR/KR]; (KR) (For US Only)
Inventors: LEE, Hyun-Joo; (KR).
KIM, Dong-Hoon; (KR).
KIM, Tae-Kyun; (KR).
YOON, Young-Ae; (KR).
SIM, Jae-Young; (KR).
CHA, Myung-Hun; (KR).
JUNG, Eun-Jung; (KR).
AHN, Kyoung-Kyu; (KR).
LEE, Tai-Au; (KR)
Agent: OH, Kook-Jin; 302, Dooeon Bldg. 1708-6, Seocho-dong, Seocho-gu Seoul 137-884 (KR)
Priority Data:
10-2011-0016981 25.02.2011 KR
Title (EN) DIAMINOPYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF
(FR) DÉRIVÉS DE DIAMINOPYRIMIDINE ET LEURS PROCÉDÉS DE PRÉPARATION
Abstract: front page image
(EN)The present invention provides a diaminopyrimidine derivative or its pharmaceutically acceptable salt, a process for the preparation thereof, a pharmaceutical composition comprising the same, and a use thereof. The diaminopyrimidine derivative or its pharmaceutically acceptable salt functions as a 5-HT4 receptor agonist, and therefore can be usefully applied for preventing or treating dysfunction in gastrointestinal motility, one of the gastrointestinal diseases, such as gastroesophageal reflux disease (GERD), constipation, irritable bowel syndrome (IBS), dyspepsia, post-operative ileus, delayed gastric emptying, gastroparesis, intestinal pseudo-obstruction, drug-induced delayed transit, or diabetic gastric atony.
(FR)Cette invention concerne un dérivé de diaminopyrimidine ou son sel de qualité pharmaceutique, un procédé pour le préparer, une composition pharmaceutique le contenant, et une de ses utilisations. Le dérivé de diaminopyrimidine ou son sel de qualité pharmaceutique agit comme un agoniste du récepteur 5-HT4 et peut, par conséquent, être appliqué de manière utile pour prévenir ou traiter le dysfonctionnement de la motilité gastro-intestinale, et une maladie gastro-intestinale telle que le reflux gastro-œsophagien (GERD), la constipation, le syndrome de l'intestin irritable (IBS), la dyspepsie, l'occlusion intestinale postopératoire, la vidange gastrique retardée, la gastroparésie, la pseudo-obstruction intestinale, le transit retardé induit par des médicaments, ou l'atonie gastrique d'origine diabétique.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: English (EN)
Filing Language: English (EN)