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1. (WO2012115446) COMPOUND BASED ON 5-(SUBSTITUTED ALKYL-AMINOMETHYL) ISOXAZOLE ACTING AS A T-TYPE CALCIUM CHANNEL ANTAGONIST
Latest bibliographic data on file with the International Bureau   

Pub. No.:    WO/2012/115446    International Application No.:    PCT/KR2012/001340
Publication Date: 30.08.2012 International Filing Date: 22.02.2012
IPC:
C07D 413/12 (2006.01), A61K 31/497 (2006.01), A61P 25/00 (2006.01), A61P 35/00 (2006.01)
Applicants: KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY [KR/KR]; 39-1 Hawolgok-dong, Seongbuk-gu Seoul 136-791 (KR) (For All Designated States Except US).
CHOO, Hyun Ah [KR/KR]; (KR) (For US Only).
PAE, Ae Nim [KR/KR]; (KR) (For US Only).
CHO, Yong Seo [KR/KR]; (KR) (For US Only).
LEE, Hyo Seon [KR/KR]; (KR) (For US Only).
LEE, Jie Eun [KR/KR]; (KR) (For US Only).
CHO, Gyeong Hi [KR/KR]; (KR) (For US Only).
RHIM, Hye Whon [KR/KR]; (KR) (For US Only).
SEO, Seon Hee [KR/KR]; (KR) (For US Only).
SONG, Chi Man [KR/KR]; (KR) (For US Only).
CHUNG, Hye Jin [KR/KR]; (KR) (For US Only).
NAM, Ghil Soo [KR/KR]; (KR) (For US Only).
KEUM, Gyo Chang [KR/KR]; (KR) (For US Only).
KIM, Dong Jin [KR/KR]; (KR) (For US Only).
CHOI, Kyung Il [KR/KR]; (KR) (For US Only).
CHOI, Kee Hyun [KR/KR]; (KR) (For US Only).
LEE, Jae Kyun [KR/KR]; (KR) (For US Only).
KANG, Yong Koo [KR/KR]; (KR) (For US Only).
PARK, Woong Seo [KR/KR]; (KR) (For US Only).
LEE, Ju Hyeon [KR/KR]; (KR) (For US Only).
SHIN, Sun Mi [KR/KR]; (KR) (For US Only).
AHMED, Abdul Waheed [PK/KR]; (KR) (For US Only).
KIM, Young Soo [KR/KR]; (KR) (For US Only).
MIN, Sun Joon [KR/KR]; (KR) (For US Only)
Inventors: CHOO, Hyun Ah; (KR).
PAE, Ae Nim; (KR).
CHO, Yong Seo; (KR).
LEE, Hyo Seon; (KR).
LEE, Jie Eun; (KR).
CHO, Gyeong Hi; (KR).
RHIM, Hye Whon; (KR).
SEO, Seon Hee; (KR).
SONG, Chi Man; (KR).
CHUNG, Hye Jin; (KR).
NAM, Ghil Soo; (KR).
KEUM, Gyo Chang; (KR).
KIM, Dong Jin; (KR).
CHOI, Kyung Il; (KR).
CHOI, Kee Hyun; (KR).
LEE, Jae Kyun; (KR).
KANG, Yong Koo; (KR).
PARK, Woong Seo; (KR).
LEE, Ju Hyeon; (KR).
SHIN, Sun Mi; (KR).
AHMED, Abdul Waheed; (KR).
KIM, Young Soo; (KR).
MIN, Sun Joon; (KR)
Agent: HALLA PATENT&LAW FIRM; 9F KAMCO Yangjae Tower 949-3 Dogok-dong, Gangnam-gu Seoul 135-270 (KR)
Priority Data:
10-2011-0016203 23.02.2011 KR
Title (EN) COMPOUND BASED ON 5-(SUBSTITUTED ALKYL-AMINOMETHYL) ISOXAZOLE ACTING AS A T-TYPE CALCIUM CHANNEL ANTAGONIST
(FR) COMPOSÉ À BASE DE 5-(ALKYLE-AMINOMÉTHYLE SUBSTITUÉ) ISOXAZOLE, AGISSANT EN TANT QU'ANTAGONISTE DU CANAL CALCIQUE DE TYPE T
(KO) T-형 칼슘 채널 길항제로서의 5-(치환된알킬아미노메틸)아이속사졸계 화합물
Abstract: front page image
(EN)The present invention relates to: a compound based on 5-(substituted alkyl-aminomethyl) isoxazole which exhibits pharmaceutical activity with respect to T-type calcium channels; a pharmaceutically acceptable salt thereof; a production method for such a compound; and to a pharmaceutical composition containing such a compound as an active ingredient.
(FR)La présente invention concerne les éléments suivants : un composé à base de 5-(alkyle-aminométhyle substitué) isoxazole présentant une activité pharmaceutique par rapport aux canaux calciques de type T ; un sel pharmaceutiquement acceptable de celui-ci ; un procédé de production d'un tel composé ; et une composition pharmaceutique contenant ledit composé en tant que principe actif.
(KO)본 발명은 T-형 칼슘 채널에 대하여 약학적 활성을 보이는 5-(치환된알킬아미노메틸)아이속사졸계 화합물 및 약제학적으로 허용 가능한 이의 염, 이들 화합물의 제조방법, 그리고 이들 화합물이 유효성분으로 함유된 약제조성물에 관한 것이다.
Designated States: AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IS, JP, KE, KG, KM, KN, KP, KZ, LA, LC, LK, LR, LS, LT, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW.
African Regional Intellectual Property Organization (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, SZ, TZ, UG, ZM, ZW)
Eurasian Patent Organization (AM, AZ, BY, KG, KZ, MD, RU, TJ, TM)
European Patent Office (AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR)
African Intellectual Property Organization (BF, BJ, CF, CG, CI, CM, GA, GN, GQ, GW, ML, MR, NE, SN, TD, TG).
Publication Language: Korean (KO)
Filing Language: Korean (KO)